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Target
Lysophosphatidic acid receptor 3
Ligand
BDBM50177338
Substrate
n/a
Meas. Tech.
ChEMBL_329846 (CHEMBL862795)
EC50
7590±n/a nM
Citation
 Gududuru, V; Zeng, K; Tsukahara, R; Makarova, N; Fujiwara, Y; Pigg, KR; Baker, DL; Tigyi, G; Miller, DD Identification of Darmstoff analogs as selective agonists and antagonists of lysophosphatidic acid receptors. Bioorg Med Chem Lett 16:451-6 (2005) [PubMed]  Article 
Target
Name:
Lysophosphatidic acid receptor 3
Synonyms:
Edg7 | LPAR3_RAT | Lpa3 | Lpar3 | Lysophosphatidic acid receptor 1/lysophosphatidic acid receptor 3 | Lysophosphatidic acid receptor Edg-7
Type:
PROTEIN
Mol. Mass.:
40307.81
Organism:
Rattus norvegicus
Description:
ChEMBL_329846
Residue:
354
Sequence:
MNECHYDKRMDFFYNRSNTDTADEWTGTKLVIVLCVGTFFCLFIFFSNSLVIAAVITNRKFHFPFYYLLANLAAADFFAGIAYVFLMFNTGPVSKTLTVNRWLLRQGLLDTSLTASLANLLVIAVERHMSIMRMRIHSNLTKKRVTLLILLVWAIAIFMGAVPTLGWNCLCNISACSSLAPIYSRSYLIFWTVSNLLAFFIMVVVYVRIYMYVKRKTNVLSPHTSGSISRRRAPMKLMKTVMTVLGAFVVCWTPGLVVLLLDGLNCKQCNVQHVKRWFLLLALLNSVMNPIIYSYKDEDMYNTMRKMICCAPHDSNAERHPSRIPSTIHSRSDTGSQYLEDSISQGQVCNKSSS
  
Inhibitor
Name:
BDBM50177338
Synonyms:
CHEMBL383362 | potassium (2-(heptadeca-9,12,15-trienyl)-1,3-dioxolan-4-yl)methyl hydrogenphosphate
Type:
Small organic molecule
Emp. Form.:
C21H36O6P
Mol. Mass.:
415.4813
SMILES:
C\C=C\C\C=C\C\C=C\CCCCCCCCC1OCC(COP(O)([O-])=O)O1
Structure:
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