Reaction Details Report a problem with these data
Target
C-C chemokine receptor type 4
Ligand
BDBM50209256
Substrate
n/a
Meas. Tech.
ChEMBL_455257 (CHEMBL906418)
Ki
10000±n/a nM
Citation
Burdi, DF; Chi, S; Mattia, K; Harrington, C; Shi, Z; Chen, S; Jacutin-Porte, S; Bennett, R; Carson, K; Yin, W; Kansra, V; Gonzalo, JA; Coyle, A; Jaffee, B; Ocain, T; Hodge, M; LaRosa, G; Harriman, G Small molecule antagonists of the CC chemokine receptor 4 (CCR4). Bioorg Med Chem Lett 17:3141-5 (2007) [PubMed] Article
More Info.:
Target
Name:
C-C chemokine receptor type 4
Synonyms:
C-C CKR-4 | C-C chemokine receptor type 4 | C-C chemokine receptor type 4 (CCR4) | CC-CKR-4 | CCR-4 | CCR4 | CCR4_HUMAN | CD_antigen=CD194 | CMKBR4 | K5-5
Type:
Enzyme
Mol. Mass.:
41406.41
Organism:
Homo sapiens (Human)
Description:
P51679
Residue:
360
Sequence:
MNPTDIADTTLDESIYSNYYLYESIPKPCTKEGIKAFGELFLPPLYSLVFVFGLLGNSVVVLVLFKYKRLRSMTDVYLLNLAISDLLFVFSLPFWGYYAADQWVFGLGLCKMISWMYLVGFYSGIFFVMLMSIDRYLAIVHAVFSLRARTLTYGVITSLATWSVAVFASLPGFLFSTCYTERNHTYCKTKYSLNSTTWKVLSSLEINILGLVIPLGIMLFCYSMIIRTLQHCKNEKKNKAVKMIFAVVVLFLGFWTPYNIVLFLETLVELEVLQDCTFERYLDYAIQATETLAFVHCCLNPIIYFFLGEKFRKYILQLFKTCRGLFVLCQYCGLLQIYSADTPSSSYTQSTMDHDLHDAL