Reaction Details Report a problem with these data
Target
Histamine H3 receptor
Ligand
BDBM22911
Substrate
n/a
Meas. Tech.
ChEMBL_86739 (CHEMBL693464)
EC50
1±n/a nM
Citation
Ganellin, CR; Bang-Andersen, B; Khalaf, YS; Tertiuk, W; Arrang, JM; Garbarg, M; Ligneau, X; Rouleau, A; Schwartz, JC Imetit and N-methyl derivatives. The transition from potent agonist to antagonist at histamine H3 receptors.1 Bioorg Med Chem Lett 2:1231-1234 (1992) Article
More Info.:
Target
Name:
Histamine H3 receptor
Synonyms:
HH3R | HRH3_RAT | Hrh3
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
48607.98
Organism:
Rattus norvegicus (rat)
Description:
n/a
Residue:
445
Sequence:
MERAPPDGLMNASGTLAGEAAAAGGARGFSAAWTAVLAALMALLIVATVLGNALVMLAFVADSSLRTQNNFFLLNLAISDFLVGAFCIPLYVPYVLTGRWTFGRGLCKLWLVVDYLLCASSVFNIVLISYDRFLSVTRAVSYRAQQGDTRRAVRKMALVWVLAFLLYGPAILSWEYLSGGSSIPEGHCYAEFFYNWYFLITASTLEFFTPFLSVTFFNLSIYLNIQRRTRLRLDGGREAGPEPPPDAQPSPPPAPPSCWGCWPKGHGEAMPLHRYGVGEAGPGVEAGEAALGGGSGGGAAASPTSSSGSSSRGTERPRSLKRGSKPSASSASLEKRMKMVSQSITQRFRLSRDKKVAKSLAIIVSIFGLCWAPYTLLMIIRAACHGRCIPDYWYETSFWLLWANSAVNPVLYPLCHYSFRRAFTKLLCPQKLKVQPHGSLEQCWK