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Target
ELAV-like protein 1
Ligand
BDBM50326010
Substrate
n/a
Meas. Tech.
ChEMBL_654856 (CHEMBL1243900)
Kd
6±n/a nM
Citation
 Meisner, NC; Hintersteiner, M; Mueller, K; Bauer, R; Seifert, JM; Naegeli, HU; Ottl, J; Oberer, L; Guenat, C; Moss, S; Harrer, N; Woisetschlaeger, M; Buehler, C; Uhl, V; Auer, M Identification and mechanistic characterization of low-molecular-weight inhibitors for HuR. Nat Chem Biol 3:508-15 (2007) [PubMed]  Article 
Target
Name:
ELAV-like protein 1
Synonyms:
ELAV1_HUMAN | ELAVL1 | HUR | Hu-antigen R
Type:
PROTEIN
Mol. Mass.:
36102.56
Organism:
Homo sapiens (Human)
Description:
ChEMBL_654855
Residue:
326
Sequence:
MSNGYEDHMAEDCRGDIGRTNLIVNYLPQNMTQDELRSLFSSIGEVESAKLIRDKVAGHSLGYGFVNYVTAKDAERAINTLNGLRLQSKTIKVSYARPSSEVIKDANLYISGLPRTMTQKDVEDMFSRFGRIINSRVLVDQTTGLSRGVAFIRFDKRSEAEEAITSFNGHKPPGSSEPITVKFAANPNQNKNVALLSQLYHSPARRFGGPVHHQAQRFRFSPMGVDHMSGLSGVNVPGNASSGWCIFIYNLGQDADEGILWQMFGPFGAVTNVKVIRDFNTNKCKGFGFVTMTNYEEAAMAIASLNGYRLGDKILQVSFKTNKSHK
  
Inhibitor
Name:
BDBM50326010
Synonyms:
CHEMBL1242196 | Dehydromutactin
Type:
Small organic molecule
Emp. Form.:
C16H12O5
Mol. Mass.:
284.2635
SMILES:
Cc1cc(O)c2c(O)cccc2c1-c1cc(O)cc(=O)o1
Structure:
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