Reaction Details Report a problem with these data
Target
Melanocortin receptor 4
Ligand
BDBM50111186
Substrate
n/a
Meas. Tech.
ChEBML_106360
Ki
>1000±n/a nM
Citation
 Mutulis, F; Mutule, I; Wikberg, JE N-alkylaminoacids and their derivatives interact with melanocortin receptors. Bioorg Med Chem Lett 12:1039-42 (2002) [PubMed]  Article 
Target
Name:
Melanocortin receptor 4
Synonyms:
MC4-R | MC4R | MC4R_HUMAN | Melanocortin MC4 | Melanocortin receptor 4 (MC-4) | Melanocortin receptor 4 (MC4-R) | Melanocortin receptor 4 (MC4R)
Type:
Enzyme
Mol. Mass.:
36949.50
Organism:
Homo sapiens (Human)
Description:
P32245
Residue:
332
Sequence:
MVNSTHRGMHTSLHLWNRSSYRLHSNASESLGKGYSDGGCYEQLFVSPEVFVTLGVISLLENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVNIDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVKRVGIIISCIWAACTVSGILFIIYSDSSAVIICLITMFFTMLALMASLYVHMFLMARLHIKRIAVLPGTGAIRQGANMKGAITLTILIGVFVVCWAPFFLHLIFYISCPQNPYCVCFMSHFNLYLILIMCNSIIDPLIYALRSQELRKTFKEIICCYPLGGLCDLSSRY
  
Inhibitor
Name:
BDBM50111186
Synonyms:
(S)-2-Benzylamino-5-guanidino-pentanoic acid amide | CHEMBL9075 | MK-27
Type:
Small organic molecule
Emp. Form.:
C13H21N5O
Mol. Mass.:
263.3387
SMILES:
NC(=N)NCCC[C@H](NCc1ccccc1)C(N)=O
Structure:
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