Reaction Details Report a problem with these data
Target
Mu-type opioid receptor
Ligand
BDBM50000781
Substrate
n/a
Meas. Tech.
ChEBML_146255
Ki
2610±n/a nM
Citation
 Cheng, CY; Wu, SC; Hsin, LW; Tam, SW Selective reversible and irreversible ligands for the kappa opioid receptor. J Med Chem 35:2243-7 (1992) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50000781
Synonyms:
2-(3,4-Dichloro-phenyl)-N-methyl-N-(3-methylene-2-oxo-8-pyrrolidin-1-yl-1-oxa-spiro[4.5]dec-7-yl)-acetamide | CHEMBL70311
Type:
Small organic molecule
Emp. Form.:
C23H28Cl2N2O3
Mol. Mass.:
451.386
SMILES:
CN([C@H]1C[C@]2(CC(=C)C(=O)O2)CC[C@@H]1N1CCCC1)C(=O)Cc1ccc(Cl)c(Cl)c1
Structure:
Search PDB for entries with ligand similarity: