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Target
Adenosine receptor A3
Ligand
BDBM50370195
Substrate
n/a
Meas. Tech.
ChEMBL_30462 (CHEMBL643123)
Ki
6160±n/a nM
Citation
 Cappellacci, L; Barboni, G; Palmieri, M; Pasqualini, M; Grifantini, M; Costa, B; Martini, C; Franchetti, P Ribose-modified nucleosides as ligands for adenosine receptors: synthesis, conformational analysis, and biological evaluation of 1'-C-methyl adenosine analogues. J Med Chem 45:1196-202 (2002) [PubMed]  Article 
Target
Name:
Adenosine receptor A3
Synonyms:
AA3R_RAT | Adenosine A3 receptor | Adenosine receptor A2a and A3 | Adora3
Type:
PROTEIN
Mol. Mass.:
36643.73
Organism:
Rattus norvegicus
Description:
ChEMBL_479910
Residue:
320
Sequence:
MKANNTTTSALWLQITYITMEAAIGLCAVVGNMLVIWVVKLNRTLRTTTFYFIVSLALADIAVGVLVIPLAIAVSLEVQMHFYACLFMSCVLLVFTHASIMSLLAIAVDRYLRVKLTVRYRTVTTQRRIWLFLGLCWLVSFLVGLTPMFGWNRKVTLELSQNSSTLSCHFRSVVGLDYMVFFSFITWILIPLVVMCIIYLDIFYIIRNKLSQNLTGFRETRAFYGREFKTAKSLFLVLFLFALCWLPLSIINFVSYFNVKIPEIAMCLGILLSHANSMMNPIVYACKIKKFKETYFVILRACRLCQTSDSLDSNLEQTTE
  
Inhibitor
Name:
BDBM50370195
Synonyms:
CHEMBL605646
Type:
Small organic molecule
Emp. Form.:
C20H25N5O4
Mol. Mass.:
399.4436
SMILES:
C[C@@H](Cc1ccccc1)Nc1ncnc2n(cnc12)C1(C)O[C@H](CO)[C@@H](O)[C@H]1O |r|
Structure:
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