Reaction Details Report a problem with these data
Target
Somatostatin receptor type 4
Ligand
BDBM50159450
Substrate
n/a
Meas. Tech.
ChEMBL_306614 (CHEMBL829074)
IC50
1±n/a nM
Citation
 Rivier, JE; Kirby, DA; Erchegyi, J; Waser, B; Eltschinger, V; Cescato, R; Reubi, JC Somatostatin receptor 1 selective analogues: 3. Dicyclic peptides. J Med Chem 48:515-22 (2005) [PubMed]  Article 
Target
Name:
Somatostatin receptor type 4
Synonyms:
SOMATOSTATIN SST4 | SS-4-R | SS4-R | SS4R | SSR4_HUMAN | SST4R | SSTR4 | Somatostatin receptor type 4 (SSTR4)
Type:
Enzyme
Mol. Mass.:
42015.38
Organism:
Homo sapiens (Human)
Description:
P31391
Residue:
388
Sequence:
MSAPSTLPPGGEEGLGTAWPSAANASSAPAEAEEAVAGPGDARAAGMVAIQCIYALVCLVGLVGNALVIFVILRYAKMKTATNIYLLNLAVADELFMLSVPFVASSAALRHWPFGSVLCRAVLSVDGLNMFTSVFCLTVLSVDRYVAVVHPLRAATYRRPSVAKLINLGVWLASLLVTLPIAIFADTRPARGGQAVACNLQWPHPAWSAVFVVYTFLLGFLLPVLAIGLCYLLIVGKMRAVALRAGWQQRRRSEKKITRLVLMVVVVFVLCWMPFYVVQLLNLFVTSLDATVNHVSLILSYANSCANPILYGFLSDNFRRFFQRVLCLRCCLLEGAGGAEEEPLDYYATALKSKGGAGCMCPPLPCQQEALQPEPGRKRIPLTRTTTF
  
Inhibitor
Name:
BDBM50159450
Synonyms:
CHEMBL386784 | Des-AA1,2,4,5,13-[D-Trp8]-SRIF
Type:
Small organic molecule
Emp. Form.:
C58H73N11O12S2
Mol. Mass.:
1180.397
SMILES:
C[C@@H](O)[C@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@H](N)CSSC[C@H](NC1=O)C(O)=O)[C@@H](C)O
Structure:
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