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Target
Mu-type opioid receptor
Ligand
BDBM50210181
Substrate
n/a
Meas. Tech.
ChEMBL_443958 (CHEMBL893119)
Ki
3320±n/a nM
Citation
 Weigl, M; Wünsch, B Synthesis of bridged piperazines with sigma receptor affinity. Eur J Med Chem 42:1247-62 (2007) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50210181
Synonyms:
6-benzyl-2-(benzyloxy)-8-butyl-6,8-diaza-bicyclo[3.2.2]nonane | CHEMBL429103
Type:
Small organic molecule
Emp. Form.:
C25H34N2O
Mol. Mass.:
378.5503
SMILES:
CCCCN1CC2CCC(OCc3ccccc3)C1CN2Cc1ccccc1 |w:18.20,9.9,6.6,TLB:3:4:20.19:7.8.9,THB:21:20:7.8.9:5.4,TEB:10:9:20.19:5.4|
Structure:
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