Reaction Details Report a problem with these data
Target
Cannabinoid receptor 2
Ligand
BDBM50396288
Substrate
n/a
Meas. Tech.
ChEMBL_863891 (CHEMBL2176375)
Ki
>1000±n/a nM
Citation
 Johnston, M; Bhatt, SR; Sikka, S; Mercier, RW; West, JM; Makriyannis, A; Gatley, SJ; Duclos, RI Assay and inhibition of diacylglycerol lipase activity. Bioorg Med Chem Lett 22:4585-92 (2012) [PubMed]  Article 
Target
Name:
Cannabinoid receptor 2
Synonyms:
CANNABINOID CB2 | CB-2 | CB2 | CNR2_MOUSE | Cannabinoid CB2 receptor | Cannabinoid receptor | Cannabinoid receptor 2 | Cnr2 | mCB2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
38220.43
Organism:
MOUSE
Description:
P47936
Residue:
347
Sequence:
MEGCRETEVTNGSNGGLEFNPMKEYMILSSGQQIAVAVLCTLMGLLSALENMAVLYIILSSRRLRRKPSYLFISSLAGADFLASVIFACNFVIFHVFHGVDSNAIFLLKIGSVTMTFTASVGSLLLTAVDRYLCLCYPPTYKALVTRGRALVALCVMWVLSALISYLPLMGWTCCPSPCSELFPLIPNDYLLGWLLFIAILFSGIIYTYGYVLWKAHRHVATLAEHQDRQVPGIARMRLDVRLAKTLGLVLAVLLICWFPALALMGHSLVTTLSDQVKEAFAFCSMLCLVNSMVNPIIYALRSGEIRSAAQHCLIGWKKYLQGLGPEGKEEGPRSSVTETEADVKTT
  
Inhibitor
Name:
BDBM50396288
Synonyms:
CHEMBL2172458
Type:
Small organic molecule
Emp. Form.:
C28H43NO4Si
Mol. Mass.:
485.7308
SMILES:
CCCCCCCCNC(=O)OCC(OC)O[Si](c1ccccc1)(c1ccccc1)C(C)(C)C
Structure:
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