Reaction Details Report a problem with these data
Target
5-hydroxytryptamine receptor 4
Ligand
BDBM50421359
Substrate
n/a
Meas. Tech.
ChEMBL_201063 (CHEMBL805839)
Ki
0.079433±n/a nM
Citation
  TBA Bioorg Med Chem Lett 4:667-668 (1994)    Article 
Target
Name:
5-hydroxytryptamine receptor 4
Synonyms:
5-hydroxytryptamine receptor 4 protein | Serotonin 4 (5-HT4) receptor
Type:
PROTEIN
Mol. Mass.:
45024.02
Organism:
Sus scrofa
Description:
ChEMBL_1297282
Residue:
402
Sequence:
MDKLDANGSSKEGFGSVEKVVLLTFVSAVILMAVLGNLLVMVAVCRDRQLRKIKTNYFIVSLAFADLLVSVLVMPFGAIELVQDVWIYGEMFCLVRTSLDVLLTTASIFHLCCISLDRYYAICCQPLVYRNKMTPLRVAVLLAGCWAIPVLISFLPIMQGWNNIGITDLERTSKPRLGQDLHVIEKRKFHQNSNSTYCIFMVNKPYAITCSVVAFYIPFLLMVLAYWRIYVTAKEHAHQIQMLQRAGAPAEGRPPSADQHSTHRMRTETKAAKTLCVIMGCFCLCWAPFFVTNVVDPFADYSVPGQVWTAFLWLGYINSGLNPFLYAFLNKSFRRAFLIILCCDDERYRRPCVAGQTVPCSTTTVNGSTHVLRDAVECGGQWESQCHPPATSPLVAAQPSDT
  
Inhibitor
Name:
BDBM50421359
Synonyms:
CHEMBL145075
Type:
Small organic molecule
Emp. Form.:
C21H28N2O3
Mol. Mass.:
356.4586
SMILES:
CCCCN1CCC(COC(=O)c2c3OCCn3c3ccccc23)CC1
Structure:
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