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Target
Platelet-activating factor receptor
Ligand
BDBM50422593
Substrate
n/a
Meas. Tech.
ChEMBL_307258 (CHEMBL830837)
IC50
2344±n/a nM
Citation
 Goldring, WP; Alexander, SP; Kendall, DA; Pattenden, G Novel phomactin analogues as PAF receptor ligands. Bioorg Med Chem Lett 15:3263-6 (2005) [PubMed]  Article 
Target
Name:
Platelet-activating factor receptor
Synonyms:
PAF Platelet activating factor | PAF-R | PAFR | PTAFR | PTAFR_HUMAN | Platelet activating factor receptor | Platelet-activating factor receptor
Type:
Enzyme Catalytic Domain
Mol. Mass.:
39219.60
Organism:
Homo sapiens (Human)
Description:
PAF Platelet activating factor PTAFR HUMAN::P25105
Residue:
342
Sequence:
MEPHDSSHMDSEFRYTLFPIVYSIIFVLGVIANGYVLWVFARLYPCKKFNEIKIFMVNLTMADMLFLITLPLWIVYYQNQGNWILPKFLCNVAGCLFFINTYCSVAFLGVITYNRFQAVTRPIKTAQANTRKRGISLSLVIWVAIVGAASYFLILDSTNTVPDSAGSGNVTRCFEHYEKGSVPVLIIHIFIVFSFFLVFLIILFCNLVIIRTLLMQPVQQQRNAEVKRRALWMVCTVLAVFIICFVPHHVVQLPWTLAELGFQDSKFHQAINDAHQVTLCLLSTNCVLDPVIYCFLTKKFRKHLTEKFYSMRSSRKCSRATTDTVTEVVVPFNQIPGNSLKN
  
Inhibitor
Name:
BDBM50422593
Synonyms:
CHEMBL363216
Type:
Small organic molecule
Emp. Form.:
C20H30O5
Mol. Mass.:
350.4492
SMILES:
C[C@@H]1C[C@H]2O[C@@]3(C)CC\C=C(C)\CC[C@@]1(C)[C@]14CO[C@](O)([C@H]3O)[C@]21O4 |c:9|
Structure:
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