Reaction Details Report a problem with these data
Target
Transmembrane protease serine 4
Ligand
BDBM50430162
Substrate
n/a
Meas. Tech.
ChEMBL_942945 (CHEMBL2343323)
IC50
85000±n/a nM
Citation
More Info.:
Target
Name:
Transmembrane protease serine 4
Synonyms:
CAPH2 | Channel-activating protease 2 | MT-SP2 | Membrane-type serine protease 2 | TMPRSS3 | TMPRSS4 | TMPS4_HUMAN
Type:
PROTEIN
Mol. Mass.:
48237.89
Organism:
Homo sapiens (Human)
Description:
ChEMBL_942945
Residue:
437
Sequence:
MLQDPDSDQPLNSLDVKPLRKPRIPMETFRKVGIPIIIALLSLASIIIVVVLIKVILDKYYFLCGQPLHFIPRKQLCDGELDCPLGEDEEHCVKSFPEGPAVAVRLSKDRSTLQVLDSATGNWFSACFDNFTEALAETACRQMGYSSKPTFRAVEIGPDQDLDVVEITENSQELRMRNSSGPCLSGSLVSLHCLACGKSLKTPRVVGVEEASVDSWPWQVSIQYDKQHVCGGSILDPHWVLTAAHCFRKHTDVFNWKVRAGSDKLGSFPSLAVAKIIIIEFNPMYPKDNDIALMKLQFPLTFSGTVRPICLPFFDEELTPATPLWIIGWGFTKQNGGKMSDILLQASVQVIDSTRCNADDAYQGEVTEKMMCAGIPEGGVDTCQGDSGGPLMYQSDQWHVVGIVSWGYGCGGPSTPGVYTKVSAYLNWIYNVWKAEL