Reaction Details Report a problem with these data
Target
Trace amine-associated receptor 1
Ligand
BDBM50096964
Substrate
n/a
Meas. Tech.
ChEMBL_1499376 (CHEMBL3583705)
EC50
1700±n/a nM
Citation
Chiellini, G; Nesi, G; Digiacomo, M; Malvasi, R; Espinoza, S; Sabatini, M; Frascarelli, S; Laurino, A; Cichero, E; Macchia, M; Gainetdinov, RR; Fossa, P; Raimondi, L; Zucchi, R; Rapposelli, S Design, Synthesis, and Evaluation of Thyronamine Analogues as Novel Potent Mouse Trace Amine Associated Receptor 1 (mTAAR1) Agonists. J Med Chem 58:5096-107 (2015) [PubMed] Article
More Info.:
Target
Name:
Trace amine-associated receptor 1
Synonyms:
TAAR1_MOUSE | Ta1 | Taar1 | Tar1 | Trace amine receptor 1 (TARR1) | Trace amine-associated receptor 1 (TAAR1) | Trace amine-associated receptor1 | Trar1
Type:
Protein
Mol. Mass.:
37635.41
Organism:
Mus musculus (Mouse)
Description:
Q923Y8
Residue:
332
Sequence:
MHLCHAITNISHRNSDWSREVQASLYSLMSLIILATLVGNLIVIISISHFKQLHTPTNWLLHSMAIVDFLLGCLIMPCSMVRTVERCWYFGEILCKVHTSTDIMLSSASIFHLAFISIDRYCAVCDPLRYKAKINISTILVMILVSWSLPAVYAFGMIFLELNLKGVEELYRSQVSDLGGCSPFFSKVSGVLAFMTSFYIPGSVMLFVYYRIYFIAKGQARSINRTNVQVGLEGKSQAPQSKETKAAKTLGIMVGVFLVCWCPFFLCTVLDPFLGYVIPPSLNDALYWFGYLNSALNPMVYAFFYPWFRRALKMVLLGKIFQKDSSRSKLFL