Reaction Details Report a problem with these data
Target
Norepinephrine transporter
Ligand
BDBM84738
Substrate
n/a
Ki
1290±n/a nM
Comments
PDSP_815
Citation
 Rothman, RB; Baumann, MH; Dersch, CM; Romero, DV; Rice, KC; Carroll, FI; Partilla, JS Amphetamine-type central nervous system stimulants release norepinephrine more potently than they release dopamine and serotonin. Synapse 39:32-41 (2001) [PubMed]  Article 
Target
Name:
Norepinephrine transporter
Synonyms:
n/a
Type:
Enzyme Catalytic Domain
Mol. Mass.:
2082.45
Organism:
RAT
Description:
Norepinephrine transporter 0 RAT::Q9JIA2
Residue:
19
Sequence:
MLLARMKPQVQPELGGADQ
  
Inhibitor
Name:
BDBM84738
Synonyms:
CAS_16105-77-4 | Fenfluramine | Fenfluramine (+) | Fenfluramine (-) | NSC_3337 | d-Fenfluramine
Type:
Small organic molecule
Emp. Form.:
C12H16F3N
Mol. Mass.:
231.2573
SMILES:
CCNC(C)Cc1cccc(c1)C(F)(F)F
Structure:
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