Reaction Details Report a problem with these data
Target
Neuropeptide Y receptor type 2
Ligand
BDBM84997
Substrate
n/a
Ki
276±n/a nM
Comments
PDSP_1373
Citation
 Goumain, M; Voisin, T; Lorinet, AM; Ducroc, R; Tsocas, A; Rozé, C; Rouet-Benzineb, P; Herzog, H; Balasubramaniam, A; Laburthe, M The peptide YY-preferring receptor mediating inhibition of small intestinal secretion is a peripheral Y(2) receptor: pharmacological evidence and molecular cloning. Mol Pharmacol 60:124-34 (2001) [PubMed]  Article 
Target
Name:
Neuropeptide Y receptor type 2
Synonyms:
NPY-Y2 | NPY2R | Neuropeptide Y receptor type 2 | Neuropeptide Y/peptide YY-Y2 receptor
Type:
Enzyme Catalytic Domain
Mol. Mass.:
42514.44
Organism:
RAT
Description:
NPY-Y2 NPY2R RAT::Q9ERC0
Residue:
381
Sequence:
MGPLGAEADENQTVEVKVELYGSGPTTPRGELPPDPEPELIDSTKLVEVQVVLILAYCSIILLGVVGNSLVIHVVIKFKSMRTVTNFFIANLAVADLLVNTLCLPFTLTYTLMGEWKMGPVLCHLVPYAQGLAVQVSTITLTVIALDRHRCIVYHLESKISKQISFLIIGLAWGVSALLASPLAIFREYSLIEIIPDFEIVACTEKWPGEEKSVYGTVYSLSTLLILYVLPLGIISFSYTRIWSKLKNHVSPGAASDHYHQRRHKTTKMLVCVVVVFAVSWLPLHAFQLAVDIDSHVLDLKEYKLIFTVFHIIAMCSTFANPLLYGWMNSNYRKAFLSAFRCEQRLDAIHSEVSMTFKAKKNLEVKKNNGLTDSFSEATNV
  
Inhibitor
Name:
BDBM84997
Synonyms:
NPY D-Trp32 | NPY D-Trp32, human, rat | NPY D-Trp32, porcine
Type:
Small organic molecule
Emp. Form.:
C196H290N56O56S
Mol. Mass.:
4358.806
SMILES:
n/a
Structure:
Search PDB for entries with ligand similarity: