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Target
Guanine nucleotide-binding protein subunit alpha-15
Ligand
BDBM34611
Substrate
n/a
IC50
>29913±n/a nM
Citation
 PubChem, PC Counterscreen for agonists of the human trace amine associated receptor 1 (TAAR1): Fluorescence-based cell-based high throughput dose response assay to identify nonselective Ga16 antagonists PubChem Bioassay (2013)[AID] 
Target
Name:
Guanine nucleotide-binding protein subunit alpha-15
Synonyms:
G protein alpha 16 | G-protein subunit alpha-16 | G-protein subunit alpha-16 (G alpha-16) | GNA15 | GNA15_HUMAN | GNA16 | Guanine nucleotide-binding protein subunit alpha-15 [Y147C]
Type:
Protein
Mol. Mass.:
43577.62
Organism:
Homo sapiens (Human)
Description:
P30679
Residue:
374
Sequence:
MARSLTWRCCPWCLTEDEKAAARVDQEINRILLEQKKQDRGELKLLLLGPGESGKSTFIKQMRIIHGAGYSEEERKGFRPLVYQNIFVSMRAMIEAMERLQIPFSRPESKHHASLVMSQDPYKVTTFEKRYAAAMQWLWRDAGIRACYERRREFHLLDSAVYYLSHLERITEEGYVPTAQDVLRSRMPTTGINEYCFSVQKTNLRIVDVGGQKSERKKWIHCFENVIALIYLASLSEYDQCLEENNQENRMKESLALFGTILELPWFKSTSVILFLNKTDILEEKIPTSHLATYFPSFQGPKQDAEAAKRFILDMYTRMYTGCVDGPEGSKKGARSRRLFSHYTCATDTQNIRKVFKDVRDSVLARYLDEINLL
  
Inhibitor
Name:
BDBM34611
Synonyms:
1-(4-bromophenyl)-3-(3-methyl-1-piperidinyl)-1-propanone;hydrochloride | 1-(4-bromophenyl)-3-(3-methylpiperidin-1-yl)propan-1-one;hydrochloride | 1-(4-bromophenyl)-3-(3-methylpiperidino)propan-1-one;hydrochloride | MLS000047942 | SMR000033942 | cid_2978552
Type:
Small organic molecule
Emp. Form.:
C15H20BrNO
Mol. Mass.:
310.229
SMILES:
CC1CCCN(CCC(=O)c2ccc(Br)cc2)C1
Structure:
Search PDB for entries with ligand similarity: