Reaction Details Report a problem with these data
Target
Matrix metalloproteinase-14 [1-20,P8S]
Ligand
BDBM120186
Substrate
n/a
Meas. Tech.
Inhibition Assay
Ki
>1000±n/a nM
Citation
 Devel, L; Beau, F; Czarny, B; Dive, V Pseudodipeptides as MMP inhibitors US Patent  US8691753 Publication Date 4/8/2014 
Target
Name:
Matrix metalloproteinase-14 [1-20,P8S]
Synonyms:
MMP-14 | MMP-X1 | MMP14 | MMP14_HUMAN | MT-MMP 1 | MT1-MMP | MT1MMP | MTMMP1 | Matrix metalloproteinase 14 | Matrix metalloproteinase-14 | Membrane-type matrix metalloproteinase 1 | Membrane-type-1 matrix metalloproteinase
Type:
Protein
Mol. Mass.:
2138.64
Organism:
Homo sapiens (Human)
Description:
Q8IXG1
Residue:
20
Sequence:
MSPAPRPSRCLLLPLLTLGT
  
Inhibitor
Name:
BDBM120186
Synonyms:
US8691753, 34
Type:
Small organic molecule
Emp. Form.:
C22H27N5O8
Mol. Mass.:
489.4785
SMILES:
Cc1nc(no1)-c1ccc(CCC(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCC(O)=O)C(N)=O)cc1 |r|
Structure:
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