Assay Method Information

Assay Name:  ChEMBL_1477936 (CHEMBL3429503)
Description:  Inhibition of C-terminal His6-tagged recombinant human membrane bound COMT expressed in Bacmid infected Sf-9 insect cells using dopamine/SAM as substrate/cofactor preincubated for 2 hrs followed by dopamine/SAM addition after 25 mins by fluorescence polarization assay
Affinity data for this assay
 

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