Assay Method Information

Assay Name:  ChEMBL_1509801 (CHEMBL3603684)
Description:  Antagonist activity at endothelin A receptor in rat A7r5 cells assessed as inhibition of ET-1-induced increase in cytosolic free Ca2+ level treated 1 min prior to ET-1 addition by fura-2 dye-based spectrofluorometric analysis
Affinity data for this assay
 

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