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Found 163 of affinity data for UniProtKB/TrEMBL: Q03311
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50377920(CHEMBL540657)
Affinity DataKi:  0.460nMAssay Description:Inhibition of mouse BuChEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50149201(3,8-DIAMINO-6-PHENYL-5-[6-[1-[2-[(1,2,3,4-TETRAHYD...)
Affinity DataKi:  0.720nMAssay Description:Inhibition of mouse BuChEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50028051(CHEMBL23626 | Diallyl-(1-phenyl-cyclohexyl)-amine)
Affinity DataKi:  500nMAssay Description:-Log (Ki) value for butyrylcholinesterase by inhibiting DFPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50028051(CHEMBL23626 | Diallyl-(1-phenyl-cyclohexyl)-amine)
Affinity DataKi:  501nMAssay Description:Displacement of [3H]5-HT binding to serotonin receptor of rat fundus membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM83449(1-(1-phenylcyclohexyl)piperidine;hydrochloride | M...)
Affinity DataKi:  520nMAssay Description:Displacement of [3H]5-HT binding to serotonin receptor of rat fundus membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM83449(1-(1-phenylcyclohexyl)piperidine;hydrochloride | M...)
Affinity DataKi:  525nMAssay Description:-Log (Ki) value for butyrylcholinesterase by inhibiting DFPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50028052(Allyl-ethyl-(1-phenyl-cyclohexyl)-amine | CHEMBL23...)
Affinity DataKi:  2.57E+3nMAssay Description:Compound was tested for serotonin receptor affinity by the displacement of [3H]- -5-HT binding to rat fundus membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50028052(Allyl-ethyl-(1-phenyl-cyclohexyl)-amine | CHEMBL23...)
Affinity DataKi:  2.60E+3nMAssay Description:-Log (Ki) value for butyrylcholinesterase by inhibiting DFPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50028053(Allyl-methyl-(1-phenyl-cyclohexyl)-amine | CHEMBL2...)
Affinity DataKi:  5.50E+3nMAssay Description:Displacement of [3H]5-HT binding to serotonin receptor of rat fundus membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50028053(Allyl-methyl-(1-phenyl-cyclohexyl)-amine | CHEMBL2...)
Affinity DataKi:  5.60E+3nMAssay Description:-Log (Ki) value for butyrylcholinesterase by inhibiting DFPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50028054(Allyl-(1-phenyl-cyclohexyl)-amine | CHEMBL281855)
Affinity DataKi:  2.69E+4nMAssay Description:Displacement of [3H]5-HT binding to serotonin receptor of rat fundus membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50028054(Allyl-(1-phenyl-cyclohexyl)-amine | CHEMBL281855)
Affinity DataKi:  2.70E+4nMAssay Description:-Log (Ki) value for butyrylcholinesterase by inhibiting DFPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50028055(CHEMBL279924 | Ethyl-(1-phenyl-cyclohexyl)-amine |...)
Affinity DataKi:  5.75E+4nMAssay Description:-Log (Ki) value for butyrylcholinesterase by inhibiting DFPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50028055(CHEMBL279924 | Ethyl-(1-phenyl-cyclohexyl)-amine |...)
Affinity DataKi:  5.80E+4nMAssay Description:Displacement of [3H]5-HT binding to serotonin receptor of rat fundus membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50312905(3alpha,8-dimethyl-1-phenethyl-1,2,3,3alpha,8,8alph...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of mouse serum BChE after 1 hr by modified Ellman's colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50467895(CHEMBL4280262)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of BuChE in Swiss Webster mouse whole blood serum using butyrylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50608266(CHEMBL5288285)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of mouse serum BuChEMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50312902(3alpha,8-dimethyl-1-phenethyl-1,2,3,3alpha,8,8alph...)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of mouse serum BChE after 1 hr by modified Ellman's colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM8963(CHEMBL32823 | Homodimeric Tacrine Analog 3b | N-[7...)
Affinity DataIC50:  9.10nMAssay Description:Inhibition of BuChE in Swiss Webster mouse whole blood serum using butyrylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM8963(CHEMBL32823 | Homodimeric Tacrine Analog 3b | N-[7...)
Affinity DataIC50:  9.10nMAssay Description:Inhibition of mouse serum BuChEMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50373109(CHEMBL406645)
Affinity DataIC50:  10nMAssay Description:Inhibition of mouse serum BChEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50014113(3alpha,8-dimethyl-1-phenethyl-1,2,3,3alpha,8,8alph...)
Affinity DataIC50:  10nMAssay Description:Inhibition of mouse serum BChE after 1 hr by modified Ellman's colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50467892(CHEMBL4283717)
Affinity DataIC50:  11nMAssay Description:Inhibition of mouse serum BuChEMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50467891(CHEMBL4279148)
Affinity DataIC50:  12nMAssay Description:Inhibition of BuChE in Swiss Webster mouse whole blood serum using butyrylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50312892(3alpha,8-dimethyl-1-phenethyl-1,2,3,3alpha,8,8alph...)
Affinity DataIC50:  14nMAssay Description:Inhibition of mouse serum BChE after 1 hr by modified Ellman's colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50312903(3alpha,8-dimethyl-1-phenethyl-1,2,3,3alpha,8,8alph...)
Affinity DataIC50:  16nMAssay Description:Inhibition of mouse serum BChE after 1 hr by modified Ellman's colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50373108(CHEMBL259523)
Affinity DataIC50:  17nMAssay Description:Inhibition of mouse serum BChEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50312904(3alpha,8-dimethyl-1-phenethyl-1,2,3,3alpha,8,8alph...)
Affinity DataIC50:  22nMAssay Description:Inhibition of mouse serum BChE after 1 hr by modified Ellman's colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50467894(CHEMBL4294287)
Affinity DataIC50:  25nMAssay Description:Inhibition of mouse serum BuChEMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50467892(CHEMBL4283717)
Affinity DataIC50:  26nMAssay Description:Inhibition of BuChE in Swiss Webster mouse whole blood serum using butyrylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50608268(CHEMBL5272055)
Affinity DataIC50:  26nMAssay Description:Inhibition of mouse serum BuChEMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50467898(CHEMBL4282214)
Affinity DataIC50:  26nMAssay Description:Inhibition of BuChE in Swiss Webster mouse whole blood serum using butyrylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50608265(CHEMBL5282048)
Affinity DataIC50:  27nMAssay Description:Inhibition of mouse serum BuChEMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50467896(CHEMBL4287068)
Affinity DataIC50:  28nMAssay Description:Inhibition of BuChE in Swiss Webster mouse whole blood serum using butyrylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50467895(CHEMBL4280262)
Affinity DataIC50:  31nMAssay Description:Inhibition of mouse serum BuChEMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50467894(CHEMBL4294287)
Affinity DataIC50:  31nMAssay Description:Inhibition of BuChE in Swiss Webster mouse whole blood serum using butyrylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50467897(CHEMBL4287482)
Affinity DataIC50:  37nMAssay Description:Inhibition of BuChE in Swiss Webster mouse whole blood serum using butyrylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50467893(CHEMBL4276832)
Affinity DataIC50:  37nMAssay Description:Inhibition of mouse serum BuChEMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50467890(CHEMBL4290902)
Affinity DataIC50:  37nMAssay Description:Inhibition of BuChE in Swiss Webster mouse whole blood serum using butyrylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50467898(CHEMBL4282214)
Affinity DataIC50:  37nMAssay Description:Inhibition of mouse serum BuChEMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM11682(2,3-dihydroxybutanedioic acid; 3-[(1S)-1-(dimethyl...)
Affinity DataIC50:  58nMAssay Description:Inhibition of mouse plasma BuChE using S-butyrylacetylthiocholine iodide as substrate measured after 30 mins by Ellman's method relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  62nMAssay Description:Inhibition of mouse serum BuChEMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50373110(CHEMBL410915)
Affinity DataIC50:  63nMAssay Description:Inhibition of mouse serum BChEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  63nMAssay Description:Inhibition of BuChE in Swiss Webster mouse whole blood serum using butyrylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50608267(CHEMBL5285687)
Affinity DataIC50:  64nMAssay Description:Inhibition of mouse serum BuChEMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50467893(CHEMBL4276832)
Affinity DataIC50:  64nMAssay Description:Inhibition of BuChE in Swiss Webster mouse whole blood serum using butyrylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50373118(CHEMBL406885)
Affinity DataIC50:  74nMAssay Description:Inhibition of mouse serum BChEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50312897(3alpha,8-dimethyl-1-phenethyl-1,2,3,3alpha,8,8alph...)
Affinity DataIC50:  79nMAssay Description:Inhibition of mouse serum BChE after 1 hr by modified Ellman's colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50312887(3alpha,8-dimethyl-1-phenethyl-1,2,3,3alpha,8,8alph...)
Affinity DataIC50:  83nMAssay Description:Inhibition of mouse serum BChE after 1 hr by modified Ellman's colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50312890(3alpha,8-dimethyl-1-phenethyl-1,2,3,3alpha,8,8alph...)
Affinity DataIC50:  97nMAssay Description:Inhibition of mouse serum BChE after 1 hr by modified Ellman's colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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