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Transformation of the Non-Selective Aminocyclohexanol-Based Hsp90 Inhibitor into a Grp94-Seletive Scaffold.
ACS Chem Biol 12: 244-253 (2017)
The University of Kansas
LSD1 Substrate Binding and Gene Expression Are Affected by HDAC1-Mediated Deacetylation.
ACS Chem Biol 12: 254-264 (2017)
Wayne State University
hBfl-1/hNOXA Interaction Studies Provide New Insights on the Role of Bfl-1 in Cancer Cell Resistance and for the Design of Novel Anticancer Agents.
ACS Chem Biol 12: 444-455 (2017)
University of California Riverside
Heat Capacity Changes for Transition-State Analogue Binding and Catalysis with Human 5'-Methylthioadenosine Phosphorylase.
ACS Chem Biol 12: 464-473 (2017)
Albert Einstein College of Medicine
An Allosteric Inhibitor Scaffold Targeting the PIF-Pocket of Atypical Protein Kinase C Isoforms.
ACS Chem Biol 12: 564-573 (2017)
Universitätsklinikum Frankfurt
Inhibition of Pax2 Transcription Activation with a Small Molecule that Targets the DNA Binding Domain.
ACS Chem Biol 12: 724-734 (2017)
University of Michigan
Ligand Discovery for a Peptide-Binding GPCR by Structure-Based Screening of Fragment- and Lead-Like Chemical Libraries.
ACS Chem Biol 12: 735-745 (2017)
Stockholm University
Structural Insights into the Inhibition of Tubulin by the Antitumor Agent 4ß-(1,2,4-triazol-3-ylthio)-4-deoxypodophyllotoxin.
ACS Chem Biol 12: 746-752 (2017)
Huazhong Agricultural University
Development of Potent, Selective SRPK1 Inhibitors as Potential Topical Therapeutics for Neovascular Eye Disease.
ACS Chem Biol 12: 825-832 (2017)
Exonate Ltd
Highly Potent Cell-Permeable and Impermeable NanoLuc Luciferase Inhibitors.
ACS Chem Biol 12: 1028-1037 (2017)
Promega Biosciences LLC
Affinity Selection-Mass Spectrometry Identifies a Novel Antibacterial RNA Polymerase Inhibitor.
ACS Chem Biol 12: 1346-1352 (2017)
Merck & Co. Inc
Fragment-Sized EthR Inhibitors Exhibit Exceptionally Strong Ethionamide Boosting Effect in Whole-Cell Mycobacterium tuberculosis Assays.
ACS Chem Biol 12: 1390-1396 (2017)
University of Cambridge
Price for Opening the Transient Specificity Pocket in Human Aldose Reductase upon Ligand Binding: Structural, Thermodynamic, Kinetic, and Computational Analysis.
ACS Chem Biol 12: 1397-1415 (2017)
Philipps-Universität Marburg
Phylogenomic Analysis of the Microviridin Biosynthetic Pathway Coupled with Targeted Chemo-Enzymatic Synthesis Yields Potent Protease Inhibitors.
ACS Chem Biol 12: 1538-1546 (2017)
University of Helsinki
Discovery and Characterization of a Eukaryotic Initiation Factor 4A-3-Selective Inhibitor That Suppresses Nonsense-Mediated mRNA Decay.
ACS Chem Biol 12: 1760-1768 (2017)
BC Cancer Agency
Efficient Inhibition of SmNACE by Coordination Complexes Is Abolished by S. mansoni Sequestration of Metal.
ACS Chem Biol 12: 1787-1795 (2017)
University of Strasburg
Small Molecule Enhancement of 20S Proteasome Activity Targets Intrinsically Disordered Proteins.
ACS Chem Biol 12: 2240-2247 (2017)
Michigan State University
Direct Interaction of Chivosazole F with Actin Elicits Cell Responses Similar to Latrunculin A but Distinct from Chondramide.
ACS Chem Biol 12: 2264-2269 (2017)
Novartis Pharma AG
Structural Basis of Analog Specificity in PKG I and II.
ACS Chem Biol 12: 2388-2398 (2017)
Baylor College of Medicine
Cell Lysate-Based AlphaLISA Deubiquitinase Assay Platform for Identification of Small Molecule Inhibitors.
ACS Chem Biol 12: 2399-2407 (2017)
University of Delaware
Synthetic Lethality Triggered by Combining Olaparib with BRCA2-Rad51 Disruptors.
ACS Chem Biol 12: 2491-2497 (2017)
Istituto Italiano di Tecnologia
Selective Targeting of Bromodomains of the Bromodomain-PHD Fingers Family Impairs Osteoclast Differentiation.
ACS Chem Biol 12: 2619-2630 (2017)
Oxford University