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Targets Binding with 12 Compounds
Target Name
Affinity Link(s)
Article(s)
UniProt
Files
17beta-hydroxysteroid dehydrogenase
IC50:
18
1
1
2D
3D
TSV
3-hydroxyacyl-CoA dehydrogenase type-2
Ki:
11
IC50:
17
Kd:
8
2
7
2D
3D
TSV
5-hydroxytryptamine receptor 1A/1B/1D/1E/1F/2A/2B/2C/3A/3B/3C/3D/3E/4/5A/6/7
Ki:
1
IC50:
15
Kd:
3
3
76
2D
3D
TSV
Aggrecan core protein
Kd:
12
1
5
2D
3D
TSV
Aldo-keto reductase family 1 member B1 [W220Y,C299A]
Ki:
12
1
9
2D
3D
TSV
Amyloid-beta precursor protein [672-711]
IC50:
12
1
25
2D
3D
TSV
AP-2 complex subunit sigma
Ki:
12
3
5
2D
3D
TSV
Aspartyl/asparaginyl beta-hydroxylase
IC50:
46
1
17
2D
3D
TSV
ATP-dependent RNA helicase DHX29
IC50:
13
6
8
2D
3D
TSV
BiP isoform A
IC50:
12
1
1
2D
3D
TSV
Bromodomain-containing protein 8
IC50:
4
Kd:
13
10
7
2D
3D
TSV
Candidapepsin-2
Ki:
1
IC50:
11
1
7
2D
3D
TSV
CB1 cannabinoid receptor-interacting protein 1
Ki:
12
2
2
2D
3D
TSV
cDNA, FLJ78895, highly similar to 3-oxo-5-alpha-steroid 4-dehydrogenase 1
IC50:
12
2
1
2D
3D
TSV
Cyclin-K/Cyclin-dependent kinase 9
IC50:
12
4
10
2D
3D
TSV
Cytochrome P450 3A1
IC50:
12
2
3
2D
3D
TSV
Cytochrome P450 4Z1
Ki:
1
IC50:
23
2
3
2D
3D
TSV
D-alanyl-D-alanine dipeptidase
Ki:
6
IC50:
6
3
1
2D
3D
TSV
Delta(7)-sterol 5(6)-desaturase
IC50:
12
1
1
2D
3D
TSV
Deoxyuridine triphosphatase, putative
Ki:
12
1
1
2D
3D
TSV
Disintegrin and metalloproteinase domain-containing protein 33
Ki:
1
IC50:
13
2
6
2D
3D
TSV
DNA polymerase alpha subunit B
Ki:
2
IC50:
10
2
1
2D
3D
TSV
DNA polymerase iota
IC50:
12
5
9
2D
3D
TSV
ELAV-like protein 1 [I180A]
IC50:
12
1
5
2D
3D
TSV
Ephrin type-A receptor 4 ligand binding domain (EphA4-LBD)
Ki:
12
Kd:
5
ITC:
1
1
6
2D
3D
TSV
Epidermal growth factor receptor [1-772,'NPH',773-1210]
IC50:
12
1
17
2D
3D
TSV
Epidermal growth factor receptor [L858R,C797S]
IC50:
12
1
16
2D
3D
TSV
Epidermal growth factor receptor/Interleukin-3
IC50:
12
1
16
2D
3D
TSV
Eyes absent homolog 3
IC50:
24
2
8
2D
3D
TSV
Gap junction alpha-1 protein
IC50:
12
1
5
2D
3D
TSV
Glycine amidinotransferase, mitochondrial
Ki:
13
7
3
2D
3D
TSV
Hemagglutinin-neuraminidase
IC50:
12
1
1
2D
3D
TSV
Histidinol dehydrogenase, chloroplastic
Ki:
4
IC50:
12
1
1
2D
3D
TSV
Histone-lysine N-methyltransferase SETDB1
IC50:
6
Kd:
9
5
8
2D
3D
TSV
Hydroxyacylglutathione hydrolase, mitochondrial
Ki:
12
4
9
2D
3D
TSV
Integrin beta
IC50:
15
1
1
2D
3D
TSV
Juvenile hormone epoxide hydrolase
IC50:
12
1
1
2D
3D
TSV
kappa-type opioid receptor isoform 1
Ki:
25
1
1
2D
3D
TSV
Linoleate 9S-lipoxygenase-4
IC50:
12
2
1
2D
3D
TSV
Low-density lipoprotein receptor-related protein 6
IC50:
13
1
3
2D
3D
TSV
Lysophospholipase-like protein 1
IC50:
12
1
6
2D
3D
TSV
Lysosomal acid lipase/cholesteryl ester hydrolase
IC50:
12
2
9
2D
3D
TSV
Methionine--tRNA ligase, mitochondrial
EC50:
12
1
6
2D
3D
TSV
Methyl-CpG-binding protein 2
IC50:
12
1
5
2D
3D
TSV
Midkine
IC50:
6
Kd:
8
3
4
2D
3D
TSV
Myocilin
Kd:
12
1
5
2D
3D
TSV
Neuronal acetylcholine receptor subunit alpha-5
Ki:
12
1
1
2D
3D
TSV
Peptidoglycan D,D-transpeptidase MrdA
IC50:
17
2
7
2D
3D
TSV
Pol polyprotein
IC50:
13
1
1
2D
3D
TSV
Potassium voltage-gated channel subfamily A member 6
IC50:
16
Kd:
1
2
4
2D
3D
TSV
Proprotein convertase subtilisin/kexin type 5
Ki:
12
3
5
2D
3D
TSV
Protein phosphatase 1 regulatory subunit 1A
IC50:
15
1
5
2D
3D
TSV
Pyruvate kinase PKLR
Ki:
16
IC50:
5
Kd:
1
4
7
2D
3D
TSV
Retinoic acid receptor alpha [200-419]
Ki:
2
Kd:
8
Other:
2
2
8
2D
3D
TSV
Rous sarcoma virus integrase
IC50:
4
EC50:
8
1
0
2D
3D
TSV
Serine protease SplB
Ki:
12
1
1
2D
3D
TSV
Small conductance calcium-activated potassium channel protein 1
Ki:
1
IC50:
9
Kd:
1
EC50:
1
9
5
2D
3D
TSV
Sodium-dependent phosphate transport protein 2C
IC50:
14
1
6
2D
3D
TSV
Sodium-dependent phosphate transporter 1
IC50:
12
1
5
2D
3D
TSV
Sodium-dependent phosphate transporter 2
IC50:
12
1
1
2D
3D
TSV
Sphingomyelinase C
Ki:
3
IC50:
12
1
1
2D
3D
TSV
Subtilisin BL
Ki:
36
1
1
2D
3D
TSV
Subtilisin Carlsberg
Ki:
11
IC50:
1
2
3
2D
3D
TSV
Suppressor of tumorigenicity 14 protein homolog
Ki:
12
1
1
2D
3D
TSV
Syndecan-2
IC50:
15
1
5
2D
3D
TSV
Transcription factor JunD
IC50:
12
1
3
2D
3D
TSV
Transcription factor SOX-18
IC50:
12
1
4
2D
3D
TSV
Tryptase gamma
Ki:
1
IC50:
9
Kd:
3
5
6
2D
3D
TSV
Ubiquitin carboxyl-terminal hydrolase 7 [208-1102]
IC50:
13
1
5
2D
3D
TSV
Virokine/NFkB inhibitor
IC50:
34
1
3
2D
3D
TSV
Zinc finger protein GLI2
IC50:
12
4
11
2D
3D
TSV