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Targets Binding with 2 Compounds
Target Name
Affinity Link(s)
Article(s)
UniProt
Files
2''-aminoglycoside nucleotidyltransferase
Ki:
2
1
4
2D
3D
TSV
3-phosphoinositide-dependent protein kinase 1 [50-359]
Kd:
2
1
7
2D
3D
TSV
3-phosphoinositide-dependent protein kinase 1 [51-359,A162V]
IC50:
2
1
8
2D
3D
TSV
3-phosphoinositide-dependent protein kinase 1 [51-359,E166D]
IC50:
2
1
8
2D
3D
TSV
3-phosphoinositide-dependent protein kinase 1 [51-359,L159M]
IC50:
2
1
8
2D
3D
TSV
3-phosphoinositide-dependent protein kinase 1 [51-359,T222A]
IC50:
2
1
8
2D
3D
TSV
3-phosphoinositide-dependent protein kinase 1 [51-359,V143T,T222A]
IC50:
2
1
9
2D
3D
TSV
3-phosphoinositide-dependent protein kinase 1 [51-359,V143T]
IC50:
2
1
8
2D
3D
TSV
4-diphosphocytidyl-2-C-methyl-D-erythritol kinase, chloroplastic/chromoplastic
IC50:
2
1
1
2D
3D
TSV
5-hydroxytryptamine receptor 2A/MAP kinase-activated protein kinase 2
IC50:
8
1
9
2D
3D
TSV
Acetate Operon Repressor (IclR)
ITC:
4
1
4
2D
3D
TSV
Acidic phospholipase A2 beta
IC50:
2
1
3
2D
3D
TSV
Actin nucleation-promoting factor WASL
IC50:
2
1
1
2D
3D
TSV
Acyl-protein thioesterase 1 [I75L,S82A,Q83P,R149H,A150R,S151A]
Ki:
2
1
9
2D
3D
TSV
Acyl-protein thioesterase 1 [I75L,S82A,Q83P]
Ki:
2
1
6
2D
3D
TSV
Acyl-protein thioesterase 1 [I75L,S82A]
Ki:
2
1
5
2D
3D
TSV
Acyl-protein thioesterase 1 [I75L]
Ki:
2
1
4
2D
3D
TSV
Acyl-protein thioesterase 1 [L176M]
Ki:
2
1
4
2D
3D
TSV
Acyl-protein thioesterase 1 [Q83P]
Ki:
2
1
4
2D
3D
TSV
Acyl-protein thioesterase 2 [H152R]
Ki:
2
1
3
2D
3D
TSV
Acyl-protein thioesterase 2 [L78I,A85S,P86Q,H152R,R153A,A154S]
Ki:
2
1
8
2D
3D
TSV
Acyl-protein thioesterase 2 [L78I,A85S,P86Q]
Ki:
2
1
5
2D
3D
TSV
Acyl-protein thioesterase 2 [L78I,A85S]
Ki:
2
1
4
2D
3D
TSV
Acyl-protein thioesterase 2 [L78I]
Ki:
2
1
3
2D
3D
TSV
Acyl-protein thioesterase 2 [M178L]
Ki:
2
1
3
2D
3D
TSV
Acyl-protein thioesterase 2 [P86Q]
Ki:
2
1
3
2D
3D
TSV
Adenylate cyclase type 1/Adenylate cyclase type 2/Adenylate cyclase type 3/Adenylate cyclase type 4/Adenylate cyclase type 5/Adenylate cyclase type 6/Adenylate cyclase type 8/Adenylyl cyclase 7
IC50:
2
2
8
2D
3D
TSV
Adenylate cyclase type 9
Ki:
2
2
10
2D
3D
TSV
Aldo-keto reductase family 1 member B1 [C299A]
Ki:
2
1
8
2D
3D
TSV
Aldose Reductase (ALR2) Mutant (L300P)
ITC:
2
1
0
2D
3D
TSV
Alkaline ceramidase 3
Ki:
2
1
5
2D
3D
TSV
Alpha-1-acid glycoprotein 1
IC50:
2
1
6
2D
3D
TSV
Alpha-2-macroglobulin
IC50:
2
1
8
2D
3D
TSV
Alpha-cobratoxin
Ki:
2
IC50:
1
1
1
2D
3D
TSV
Alpha-fucosidase-like protein
Kd:
8
ITC:
8
1
1
2D
3D
TSV
Alpha-N-acetylgalactosaminide alpha-2,6-sialyltransferase 3
Ki:
2
1
1
2D
3D
TSV
Aminodeoxyfutalosine synthase
Ki:
1
IC50:
2
1
1
2D
3D
TSV
AN1-type domain-containing protein
IC50:
2
1
1
2D
3D
TSV
Androgen-dependent TFPI-regulating protein
IC50:
2
1
5
2D
3D
TSV
Androgen-induced gene 1 protein
IC50:
2
1
10
2D
3D
TSV
Apamin
Ki:
2
2
1
2D
3D
TSV
Apical membrane antigen 1
Kd:
4
1
1
2D
3D
TSV
Arginine--tRNA ligase, cytoplasmic
IC50:
2
1
5
2D
3D
TSV
Arylamine N-acetyltransferase
IC50:
8
1
2
2D
3D
TSV
Aspartate-semialdehyde dehydrogenase
IC50:
2
1
1
2D
3D
TSV
ATP-dependent RNA helicase DDX39A
IC50:
2
1
6
2D
3D
TSV
ATP-dependent translocase ABCB1 bd-verapamil
IC50:
2
1
2
2D
3D
TSV
ATP-dependent translocase ABCB1 bd-vinblastine
IC50:
2
1
2
2D
3D
TSV
ATP-diphosphohydrolase 1
IC50:
2
1
1
2D
3D
TSV
Aurora kinase C/Inner centromere protein
Ki:
1
IC50:
1
2
9
2D
3D
TSV
Beta-1,3-galactosyltransferase 1
IC50:
3
1
4
2D
3D
TSV
Beta-lactamase [1-20]
IC50:
2
1
3
2D
3D
TSV
Beta-lactamase [24-383]
Ki:
2
Kd:
2
ITC:
2
1
1
2D
3D
TSV
Beta-lactoglobulin
Kd:
2
1
3
2D
3D
TSV
Beta-xylosidase
Ki:
2
1
1
2D
3D
TSV
BH3-interacting domain death agonist [79-99]
IC50:
2
1
6
2D
3D
TSV
Bifunctional cytochrome P450/NADPH--P450 reductase [A82F,F87V]
Kd:
2
1
5
2D
3D
TSV
Bifunctional cytochrome P450/NADPH--P450 reductase [A82F]
Kd:
2
1
4
2D
3D
TSV
Bifunctional cytochrome P450/NADPH--P450 reductase [F87V]
Kd:
2
1
4
2D
3D
TSV
Bifunctional UDP-N-acetylglucosamine 2-epimerase/N-acetylmannosamine kinase
Kd:
2
1
12
2D
3D
TSV
Botulinum neurotoxin type B
IC50:
2
1
3
2D
3D
TSV
Breast cancer type 2 susceptibility protein/DNA repair protein RAD51 homolog 1
EC50:
2
1
11
2D
3D
TSV
Bromodomain-containing protein 4 [44-166,D144A]
Kd:
4
1
7
2D
3D
TSV
Bromodomain-containing protein 4 [44-166,D145A]
Kd:
4
1
7
2D
3D
TSV
Bromodomain-containing protein 4 [44-166,I246A]
Kd:
4
1
7
2D
3D
TSV
Bromodomain-containing protein 4 [44-166,L94A]
Kd:
4
1
7
2D
3D
TSV
Bromodomain-containing protein 4 [44-166,M149A]
Kd:
3
1
7
2D
3D
TSV
Bromodomain-containing protein 4 [44-166,P82A]
Kd:
4
1
7
2D
3D
TSV
Bromodomain-containing protein 4 [44-166,W81A]
Kd:
3
1
7
2D
3D
TSV
Bromodomain-containing protein 4 [44-166,Y139F]
Kd:
4
1
7
2D
3D
TSV
Bromodomain-containing protein 4 [44-166]
Kd:
4
1
6
2D
3D
TSV
CAAX prenyl protease 1 homolog
IC50:
2
1
4
2D
3D
TSV
Calcineurin subunit B type 1
IC50:
2
1
8
2D
3D
TSV
Cannabinoid receptor 1 [D338A]
Kd:
2
1
11
2D
3D
TSV
Cannabinoid receptor 1 [H219A]
Kd:
2
1
11
2D
3D
TSV
Cannabinoid receptor 1 [I218A]
Kd:
2
1
11
2D
3D
TSV
Cannabinoid receptor 1 [I339A]
Kd:
2
1
11
2D
3D
TSV
Cannabinoid receptor 1 [I341A]
Kd:
2
1
11
2D
3D
TSV
Cannabinoid receptor 1 [P221A]
Kd:
2
1
11
2D
3D
TSV
Cannabinoid receptor 1 [R340A]
Kd:
2
1
11
2D
3D
TSV
Cannabinoid receptor 1 [T344A]
Kd:
2
1
11
2D
3D
TSV
Carbon monoxide dehydrogenase small chain
Kd:
2
1
4
2D
3D
TSV
Casein kinase I
Kd:
4
1
4
2D
3D
TSV
Cdc2
IC50:
4
1
1
2D
3D
TSV
Cell division control protein 42 homolog/Ras-related C3 botulinum toxin substrate 1
IC50:
2
1
11
2D
3D
TSV
Cell division protein ZipA
Ki:
1
Kd:
2
2
1
2D
3D
TSV
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3B [654-1073]
IC50:
2
1
6
2D
3D
TSV
Chitooligosaccharidolytic beta-N-acetylglucosaminidase
Ki:
2
1
1
2D
3D
TSV
Chorismatase
Ki:
2
IC50:
2
1
1
2D
3D
TSV
Complement decay-accelerating factor
EC50:
2
1
13
2D
3D
TSV
Cone cGMP-specific 3',5'-cyclic phosphodiesterase subunit alpha'/cGMP-specific 3',5'-cyclic phosphodiesterase
Ki:
4
1
11
2D
3D
TSV
Coproheme decarboxylase
Kd:
3
1
1
2D
3D
TSV
Corticotropin releasing hormone receptor 2
IC50:
2
1
1
2D
3D
TSV
COUP transcription factor 1
IC50:
2
2
1
2D
3D
TSV
Cyclic AMP receptor protein
IC50:
2
1
1
2D
3D
TSV
Cyclin-A2 [171-432]/Cyclin-dependent kinase 2 [F82H,L83V,H84D,K98T]
IC50:
2
1
11
2D
3D
TSV
Cyclin-A2 [171-432]/Cyclin-dependent kinase 2 [F82H,L83V,H84D]
IC50:
2
1
10
2D
3D
TSV
Cyclin-A2 [171-432]/Cyclin-dependent kinase 2 [K89T]
IC50:
2
1
8
2D
3D
TSV
Cyclin-dependent kinase 2 [A144G]
IC50:
2
1
4
2D
3D
TSV
Cyclin-dependent kinase 2 [C118I]
IC50:
2
1
4
2D
3D
TSV
Cyclin-dependent kinase 2 [F80M]
IC50:
2
1
4
2D
3D
TSV
Cyclin-dependent kinase 2 [F80T]
IC50:
2
1
4
2D
3D
TSV
Cyclin-dependent protein kinase 2 variant (CDK2 A144C)
IC50:
2
Kd:
1
ITC:
1
1
4
2D
3D
TSV
Cyclin-dependent protein kinase 2 variant (CDK2 C118L)
IC50:
2
Kd:
1
ITC:
1
1
4
2D
3D
TSV
Cyclin-dependent protein kinase 2 variant (CDK2 C118L/A144C)
IC50:
2
Kd:
1
ITC:
1
1
5
2D
3D
TSV
Cyclin-dependent protein kinase PHO85
IC50:
2
1
5
2D
3D
TSV
Cytochrome c oxidase subunit NDUFA4
IC50:
4
1
4
2D
3D
TSV
Cytochrome P450 165B3
Kd:
2
1
1
2D
3D
TSV
Cytochrome P450 2B4 Mutant (F206A)
ITC:
2
1
0
2D
3D
TSV
Cytochrome P450 3A43
IC50:
2
2
9
2D
3D
TSV
Cytochrome P450 4F12
IC50:
4
1
6
2D
3D
TSV
Cytochrome P450 4F3
IC50:
8
1
5
2D
3D
TSV
Cytochrome P450 4F8
IC50:
4
1
1
2D
3D
TSV
D-3-phosphoglycerate dehydrogenase [3-314]
IC50:
2
1
5
2D
3D
TSV
D-alanine--D-alanine ligase B
IC50:
2
1
1
2D
3D
TSV
D-alanyl-D-alanine carboxypeptidase DacA
Ki:
2
1
1
2D
3D
TSV
D-aspartate oxidase 1
EC50:
2
1
1
2D
3D
TSV
D-aspartate oxidase 2
EC50:
2
1
4
2D
3D
TSV
D-aspartate oxidase 3
EC50:
2
1
3
2D
3D
TSV
D-beta-D-heptose 7-phosphate kinase
IC50:
2
1
1
2D
3D
TSV
DCN1-like protein 2
Ki:
2
2
7
2D
3D
TSV
DCN1-like protein 3
Ki:
2
2
3
2D
3D
TSV
DCN1-like protein 4
Ki:
2
2
5
2D
3D
TSV
DCN1-like protein 5
Ki:
2
2
3
2D
3D
TSV
Dihydrofolate reductase [F98Y]
Ki:
2
IC50:
2
1
3
2D
3D
TSV
Dimer of Gag-Pol polyprotein [501-599,Q508K,L534I,L564I,C568A,C596A,I585V]
Ki:
2
1
7
2D
3D
TSV
Dimer of Gag-Pol polyprotein [501-599,Q508K,L534I,L564I,C568A,C596A,L591M]
Ki:
2
1
7
2D
3D
TSV
Dimer of Gag-Pol polyprotein [501-599,Q508K,L534I,L564I,C568A,C596A,V583A]
Ki:
2
1
7
2D
3D
TSV
DNA (cytosine-5)-methyltransferase 1 [621-1600]
IC50:
3
1
7
2D
3D
TSV
DNA ligase 3
IC50:
2
1
6
2D
3D
TSV
DNA(calf thymus)
ITC:
2
1
0
2D
3D
TSV
DNA-dependent protein kinase catalytic subunit/Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
IC50:
2
1
12
2D
3D
TSV
DNA-dependent protein kinase catalytic subunit/Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
IC50:
2
1
14
2D
3D
TSV
DNA-dependent protein kinase catalytic subunit/Serine/threonine-protein kinase mTOR
IC50:
2
1
15
2D
3D
TSV
DNA-directed RNA polymerase subunit beta [D516V]
IC50:
2
1
1
2D
3D
TSV
DNA-directed RNA polymerase subunit beta [H526D]
IC50:
2
1
1
2D
3D
TSV
DNA-directed RNA polymerase subunit beta [S531L]
IC50:
2
1
1
2D
3D
TSV
DNA-directed RNA polymerase, mitochondrial
IC50:
2
2
3
2D
3D
TSV
DnaJ homolog subfamily A member 1
EC50:
2
1
4
2D
3D
TSV
Dual specificity protein kinase CLK1/CLK4
IC50:
8
1
5
2D
3D
TSV
Dual specificity protein phosphatase 15
IC50:
2
1
10
2D
3D
TSV
Dual specificity protein phosphatase 5
IC50:
19
1
4
2D
3D
TSV
Ecdysone receptor/Ultraspiracle protein
Ki:
3
IC50:
1
1
8
2D
3D
TSV
Endochitinase B1 [Y245F]
Kd:
2
2
3
2D
3D
TSV
Epidermal growth factor receptor substrate 15
IC50:
1
Kd:
1
2
5
2D
3D
TSV
Epidermal growth factor receptor [1-745,751-1210,T790M]
IC50:
2
1
17
2D
3D
TSV
Epidermal growth factor receptor [1-746,750-1210,A750P]
IC50:
2
1
17
2D
3D
TSV
Epidermal growth factor receptor [1-746,753-1210,P753S]
IC50:
2
1
17
2D
3D
TSV
Epidermal growth factor receptor [1-751,75360-1210]
IC50:
2
1
16
2D
3D
TSV
Epidermal growth factor receptor [696-1022,G719S]
Kd:
2
1
16
2D
3D
TSV
Epidermal growth factor receptor [696-1022,T790M,L858R]
Kd:
2
1
17
2D
3D
TSV
Epidermal growth factor receptor [696-1022,T790M]
Kd:
2
1
16
2D
3D
TSV
Epididymis-specific alpha-mannosidase
IC50:
2
1
4
2D
3D
TSV
Exo-1,5-alpha-L-arabinofuranobiosidase
Ki:
4
1
1
2D
3D
TSV
Exopolyphosphatase PRUNE1
IC50:
2
1
12
2D
3D
TSV
F420-dependent glucose-6-phosphate dehydrogenase
Kd:
2
1
5
2D
3D
TSV
F420-dependent glucose-6-phosphate dehydrogenase [E109Q]
Kd:
2
1
5
2D
3D
TSV
F420-dependent glucose-6-phosphate dehydrogenase [H40A]
Kd:
2
1
5
2D
3D
TSV
F420-dependent glucose-6-phosphate dehydrogenase [W44A]
Kd:
2
1
5
2D
3D
TSV
F420-dependent glucose-6-phosphate dehydrogenase [W44F]
Kd:
2
1
5
2D
3D
TSV
F420-dependent glucose-6-phosphate dehydrogenase [W44Y]
Kd:
2
1
5
2D
3D
TSV
Fatty acid-binding protein 5-ANS
Kd:
2
1
1
2D
3D
TSV
Forkhead box protein M1
Ki:
2
IC50:
2
1
7
2D
3D
TSV
Forkhead box protein O1
IC50:
2
1
5
2D
3D
TSV
Frequenin 2, isoform D
Kd:
2
1
1
2D
3D
TSV
G protein-coupled receptor 119
EC50:
2
2
4
2D
3D
TSV
Gag-Pol polyprotein [588-1147,K652R,M771V]
IC50:
2
1
6
2D
3D
TSV
Gag-Pol polyprotein [588-1147,M628L,N654N,K657R,T802F,K807E]
IC50:
2
1
9
2D
3D
TSV
Gag-Pol polyprotein [588-1147,M628L,T656S,M771V,L797W,T802Y]
IC50:
2
1
9
2D
3D
TSV
Gag-Pol polyprotein [588-1147,V662I,F664L,F703Y,Q738M,M771V]
IC50:
2
1
9
2D
3D
TSV
Gag-Pol polyprotein [600-1028,D666N,K669R,T814F,K818Q,C879S]/[600-1151,D666N,K669R,T814F,K818Q,C879S]
IC50:
1
1
9
2D
3D
TSV
Gag-Pol polyprotein [600-1028,L699I,K702N,C879S]/[600-1151,L699I,K702N,C879S]
IC50:
1
1
7
2D
3D
TSV
Gag-Pol polyprotein [600-1028,V705A,Y780C,C879S]/[600-1151,V705A,Y780C,C879S]
IC50:
1
1
7
2D
3D
TSV
Gag-Pol polyprotein [600-1028,Y780C]/[600-1151,Y780C]
IC50:
1
1
5
2D
3D
TSV
Gag-Pol polyprotein [600-1028,Y787L]/[600-1151,Y787L]
IC50:
1
1
5
2D
3D
TSV
Gag-Pol polyprotein [A1275T]
IC50:
4
1
1
2D
3D
TSV
Galactocerebrosidase
Ki:
2
1
4
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1/beta-3
EC50:
2
2
15
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1/beta-3/delta
EC50:
2
1
6
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-6/beta-2
IC50:
2
1
3
2D
3D
TSV
Gamma-enolase
IC50:
2
1
4
2D
3D
TSV
Gamma-secretase-activating protein
IC50:
2
1
7
2D
3D
TSV
Genome polyprotein [1027-1206,R1052K]
Ki:
2
Koff:
2
Kon:
2
1
2
2D
3D
TSV
Genome polyprotein [1517-1688]/Mastoparan-2 [1420-1466]
IC50:
2
Kd:
2
1
2
2D
3D
TSV
Genome polyprotein [2420-2989,M2833T,R2963Q]
IC50:
2
1
3
2D
3D
TSV
Genome polyprotein [2420-2989,M2842K,R2963Q]
IC50:
2
1
3
2D
3D
TSV
Genome polyprotein [2420-2989,P2914A,R2963Q]
IC50:
2
1
3
2D
3D
TSV
Genome polyprotein [2420-2989,R2920E,R2963Q]
IC50:
2
1
3
2D
3D
TSV
GlpG protein
IC50:
2
1
1
2D
3D
TSV
Glutathione-disulfide reductase
Ki:
2
IC50:
2
1
3
2D
3D
TSV
Gonadotropin releasing hormone receptor
IC50:
2
1
1
2D
3D
TSV
Gonadotropin-releasing hormone II receptor
IC50:
2
1
1
2D
3D
TSV
Granulocyte colony-stimulating factor receptor
Kd:
2
1
1
2D
3D
TSV
Group XIIB secretory phospholipase A2-like protein
IC50:
6
2
5
2D
3D
TSV
Guanine nucleotide binding protein, alpha q polypeptide
IC50:
2
1
1
2D
3D
TSV
H1/H5-depleted chromatin
ITC:
2
1
7
2D
3D
TSV
Histidine protein kinase SaeS
IC50:
2
Kd:
2
1
3
2D
3D
TSV
Histone acetyltransferase KAT7
IC50:
2
2
9
2D
3D
TSV
Histone acetyltransferase type B catalytic subunit
IC50:
2
2
7
2D
3D
TSV
Histone deacetylase 3/Nuclear receptor corepressor 1
IC50:
2
2
11
2D
3D
TSV
Histone deacetylase 6 [25-831]
IC50:
2
1
1
2D
3D
TSV
Histone deacetylase 6 [60-420]
Ki:
1
IC50:
1
Kd:
1
1
1
2D
3D
TSV
Histone deacetylase 6 [84-835]
Ki:
1
IC50:
1
Kd:
1
1
6
2D
3D
TSV
Histone-lysine N-methyltransferase 2B
IC50:
2
2
9
2D
3D
TSV
Histone-lysine N-methyltransferase 2D
IC50:
2
2
3
2D
3D
TSV
Histone-lysine N-methyltransferase EZH2 [Y641H]
IC50:
2
1
10
2D
3D
TSV
Histone-lysine N-methyltransferase EZH2 [Y641N]
IC50:
2
1
10
2D
3D
TSV
Histone-lysine N-methyltransferase EZH2 [Y641S]
IC50:
2
1
10
2D
3D
TSV
Histone-lysine N-methyltransferase SETD1B
IC50:
2
2
3
2D
3D
TSV
HLA class II histocompatibility antigen gamma chain/Proto-oncogene tyrosine-protein kinase ROS
IC50:
2
1
13
2D
3D
TSV
Hydroxymethylglutaryl-CoA synthase, cytoplasmic
IC50:
2
1
1
2D
3D
TSV
Hydroxysteroid 11-beta dehydrogenase 1
Ki:
1
IC50:
2
2
1
2D
3D
TSV
IGF-like family receptor 1
IC50:
1
Kd:
1
2
3
2D
3D
TSV
Immunoglobulin A1 protease autotransporter
IC50:
2
1
1
2D
3D
TSV
Inactive phospholipase C-like protein 1
IC50:
3
1
1
2D
3D
TSV
Inositol 1,4,5-trisphosphate receptor type 1/2/3
Ki:
1
EC50:
3
1
10
2D
3D
TSV
Inositol-tetrakisphosphate 1-kinase
Ki:
2
2
4
2D
3D
TSV
Insulin-like growth factor-binding protein 1
Ki:
2
1
5
2D
3D
TSV
Insulin-like growth factor-binding protein 2
Ki:
2
1
4
2D
3D
TSV
Insulin-like growth factor-binding protein 4
Ki:
2
1
6
2D
3D
TSV
Insulin-like growth factor-binding protein 6
Ki:
2
1
3
2D
3D
TSV
Integrin beta-7
IC50:
2
1
4
2D
3D
TSV
Interferon gamma receptor 1
IC50:
2
1
5
2D
3D
TSV
Interleukin 1 receptor associated kinase 4
IC50:
2
1
1
2D
3D
TSV
Interleukin-6 receptor subunit alpha
Ki:
2
1
1
2D
3D
TSV
Intracellular chorismate mutase
IC50:
2
1
5
2D
3D
TSV
Iodotyrosine deiodinase 1 [1-1,32-289]
Kd:
2
1
12
2D
3D
TSV
Isocitrate dehydrogenase [NADP] cytoplasmic [R132G]
IC50:
2
1
8
2D
3D
TSV
Isocitrate dehydrogenase [NADP], mitochondrial [R172S]
IC50:
2
1
5
2D
3D
TSV
Isoform 1 of Misshapen-like kinase 1 (MINK-delta)
IC50:
2
1
7
2D
3D
TSV
Isoform 2 of Tyrosine-protein kinase Fyn (T)
IC50:
2
1
9
2D
3D
TSV
Isoform PDE2A1 of cGMP-dependent 3',5'-cyclic phosphodiesterase (PDE2A1)
IC50:
3
2
10
2D
3D
TSV
Isoform PNNOS of Nitric oxide synthase, brain (PNNOS) -973,I269V,H341L]
Kd:
2
1
5
2D
3D
TSV
Kinesin-1 heavy chain
IC50:
2
2
4
2D
3D
TSV
Kinesin-like protein KIF20B
IC50:
8
1
23
2D
3D
TSV
Kinesin-like protein KIF23
IC50:
2
2
4
2D
3D
TSV
Kv channel-interacting protein 2/Potassium voltage-gated channel subfamily D member 3
IC50:
2
2
26
2D
3D
TSV
L-ornithine N(5)-monooxygenase
IC50:
2
Kd:
2
2
4
2D
3D
TSV
Laccase
IC50:
6
1
1
2D
3D
TSV
LanC-like protein 2
IC50:
1
Kd:
1
2
6
2D
3D
TSV
Lanosterol 14-alpha demethylase [F78L]
Kd:
2
1
5
2D
3D
TSV
Long-chain fatty acid transport protein 2
IC50:
2
1
5
2D
3D
TSV
Lymphocyte antigen 96/Toll-like receptor 4
IC50:
1
Kd:
1
2
20
2D
3D
TSV
Lysine decarboxylase
Ki:
2
1
1
2D
3D
TSV
Macrophage mannose receptor 1
IC50:
2
1
5
2D
3D
TSV
Macrophage-stimulating protein receptor [983-1400,G1195S]
IC50:
2
1
8
2D
3D
TSV
Major capsid protein L1
IC50:
2
Kd:
1
1
3
2D
3D
TSV
Mast/stem cell growth factor receptor Kit [1-973]
IC50:
2
1
9
2D
3D
TSV
Matrix metalloproteinase-19
IC50:
2
1
6
2D
3D
TSV
Matrix metalloproteinase-20
Ki:
1
IC50:
1
2
3
2D
3D
TSV
Mediator of RNA polymerase II transcription subunit 15
Ki:
1
IC50:
1
Kd:
1
1
1
2D
3D
TSV
Meiotic mRNA stability protein kinase SSN3
IC50:
2
1
3
2D
3D
TSV
Membrane-associated progesterone receptor component 1
Ki:
2
1
4
2D
3D
TSV
Metabotropic glutamate receptor 2/3
Ki:
2
EC50:
1
1
2
2D
3D
TSV
Methylcytosine dioxygenase TET3
IC50:
2
1
7
2D
3D
TSV
Mitochondrial 2-oxodicarboxylate carrier
IC50:
2
1
5
2D
3D
TSV
Mitochondrial pyruvate carrier 2
IC50:
2
1
5
2D
3D
TSV
Mitogen-activated protein kinase kinase kinase 21
IC50:
3
3
10
2D
3D
TSV
Monocarboxylate transporter 10
Ki:
2
1
3
2D
3D
TSV
Mu-type opioid/Nociceptin receptor
EC50:
4
1
12
2D
3D
TSV
Muscarinic acetylcholine receptor M3 [1-273,470-589,N6Q,N15Q,N41Q,N48Q,N52Q,A177C]
Ki:
1
Kd:
1
1
10
2D
3D
TSV
Muscarinic acetylcholine receptor M3 [1-273,470-589,N6Q,N15Q,N41Q,N48Q,N52Q,F550C]
Ki:
2
Kd:
2
1
10
2D
3D
TSV
Muscarinic acetylcholine receptor M3 [1-273,470-589,N6Q,N15Q,N41Q,N48Q,N52Q,F554C]
Ki:
1
Kd:
1
1
10
2D
3D
TSV
Muscarinic acetylcholine receptor M3 [1-273,470-589,N6Q,N15Q,N41Q,N48Q,N52Q,K178C]
Ki:
1
Kd:
1
1
10
2D
3D
TSV
Muscarinic acetylcholine receptor M3 [1-273,470-589,N6Q,N15Q,N41Q,N48Q,N52Q,K548C]
Ki:
1
Kd:
1
1
10
2D
3D
TSV
Muscarinic acetylcholine receptor M3 [1-273,470-589,N6Q,N15Q,N41Q,N48Q,N52Q,K555C]
Ki:
1
Kd:
1
1
10
2D
3D
TSV
Muscarinic acetylcholine receptor M3 [1-273,470-589,N6Q,N15Q,N41Q,N48Q,N52Q,R176C]
Ki:
2
Kd:
2
1
10
2D
3D
TSV
Muscarinic acetylcholine receptor M3 [1-273,470-589,N6Q,N15Q,N41Q,N48Q,N52Q,R179C]
Ki:
1
Kd:
1
1
10
2D
3D
TSV
Muscarinic acetylcholine receptor M3 [1-273,470-589,N6Q,N15Q,N41Q,N48Q,N52Q,R551C]
Ki:
1
Kd:
1
1
10
2D
3D
TSV
Muscarinic acetylcholine receptor M3 [1-273,470-589,N6Q,N15Q,N41Q,N48Q,N52Q,T180C]
Ki:
2
Kd:
2
1
10
2D
3D
TSV
Muscarinic acetylcholine receptor M3 [1-273,470-589,N6Q,N15Q,N41Q,N48Q,N52Q,T549C]
Ki:
1
Kd:
1
1
10
2D
3D
TSV
Muscarinic acetylcholine receptor M3 [1-273,470-589,N6Q,N15Q,N41Q,N48Q,N52Q,T552C]
Ki:
1
Kd:
1
1
10
2D
3D
TSV
Muscarinic acetylcholine receptor M3 [1-273,470-589,N6Q,N15Q,N41Q,N48Q,N52Q,T553C]
Ki:
2
Kd:
2
1
10
2D
3D
TSV
Muscarinic acetylcholine receptor M3 [1-273,470-589,N6Q,N15Q,N41Q,N48Q,N52Q,T556C]
Ki:
2
Kd:
2
1
10
2D
3D
TSV
Muscarinic acetylcholine receptor M3 [1-273,470-589,N6Q,N15Q,N41Q,N48Q,N52Q]
Ki:
3
Kd:
3
1
9
2D
3D
TSV
Myelin transcription factor 1
IC50:
2
1
7
2D
3D
TSV
Myeloid differentiation primary response protein MyD88
Kd:
2
1
11
2D
3D
TSV
Myosin-4
IC50:
2
1
3
2D
3D
TSV
N-acetyllactosaminide beta-1,3-N-acetylglucosaminyltransferase 3
Ki:
4
1
7
2D
3D
TSV
NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 11
IC50:
2
1
3
2D
3D
TSV
Neuronal calcium sensor 1
Kd:
2
1
5
2D
3D
TSV
Nitric oxide synthase oxygenase [E25A,E26A,E316A]
IC50:
2
1
3
2D
3D
TSV
Nitric oxide synthase oxygenase [E25A,E26A,I218V,E316A]
IC50:
2
1
4
2D
3D
TSV
Nitric oxide synthase, endothelial [1-973,L111A]
Kd:
2
1
2
2D
3D
TSV
Nitric oxide synthase, endothelial [1-973,Y477A]
Kd:
2
1
2
2D
3D
TSV
NS5B
IC50:
8
2
1
2D
3D
TSV
Nuclear receptor REV-ERBβ ligand-binding domain (REV-ERBβ-LBD)
ITC:
2
1
5
2D
3D
TSV
Nuclear receptor subfamily 4 group A member 3
IC50:
2
1
10
2D
3D
TSV
Nucleophosmin
EC50:
2
1
23
2D
3D
TSV
Nucleoprotein TPR
IC50:
2
1
4
2D
3D
TSV
Ovarian cancer G-protein coupled receptor 1
IC50:
2
2
5
2D
3D
TSV
Oxysterol-binding protein 2
Kd:
2
1
12
2D
3D
TSV
Oxysterol-binding protein 2 [1-181,275-916]
Kd:
2
1
13
2D
3D
TSV
p-hydroxybenzoate hydroxylase
Ki:
2
IC50:
1
1
1
2D
3D
TSV
Palmitoyl-protein thioesterase 1
IC50:
2
1
4
2D
3D
TSV
Pantothenate kinase 1, putative
IC50:
2
1
1
2D
3D
TSV
Peptidyl-prolyl cis-trans isomerase FKBP3
Ki:
2
2
4
2D
3D
TSV
Peptidyl-prolyl cis-trans isomerase H
Ki:
2
1
3
2D
3D
TSV
Peptidyl-prolyl cis-trans isomerase Mip
Ki:
2
1
1
2D
3D
TSV
Peptidyl-prolyl cis-trans isomerase-like 1
Ki:
2
1
4
2D
3D
TSV
Peripheral-type benzodiazepine receptor-associated protein 1
Ki:
2
2
4
2D
3D
TSV
Peroxisomal carnitine O-octanoyltransferase
IC50:
3
1
7
2D
3D
TSV
Pgap1 family protein
EC50:
2
1
1
2D
3D
TSV
Phosphatidylglycerophosphatase and protein-tyrosine phosphatase 1
IC50:
2
1
6
2D
3D
TSV
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform/Serine/threonine-protein kinase mTOR
IC50:
2
1
9
2D
3D
TSV
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha/delta isoform
IC50:
2
1
8
2D
3D
TSV
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform/Serine/threonine-protein kinase mTOR
IC50:
2
1
11
2D
3D
TSV
Phosphoinositide 3-kinase regulatory subunit 4
IC50:
2
2
3
2D
3D
TSV
Plasma alpha-L-fucosidase
Ki:
2
1
6
2D
3D
TSV
Platelet-derived growth factor receptor alpha [1-973]
IC50:
2
1
7
2D
3D
TSV
Platelet-derived growth factor subunit A
Ki:
1
IC50:
1
2
4
2D
3D
TSV
Pleiotrophin
Kd:
4
1
5
2D
3D
TSV
Polyketide synthase Pks13
IC50:
2
2
1
2D
3D
TSV
Polyprotein P1234
EC50:
2
1
1
2D
3D
TSV
Porphobilinogen deaminase
Ki:
2
1
7
2D
3D
TSV
Potassium channel subfamily K member 4
EC50:
2
2
4
2D
3D
TSV
POU domain, class 2, transcription factor 1
IC50:
3
2
10
2D
3D
TSV
Presequence protease, mitochondrial
EC50:
6
1
14
2D
3D
TSV
Pro-epidermal growth factor
Ki:
2
2
8
2D
3D
TSV
Probable ATP-dependent RNA helicase DDX17
IC50:
2
1
6
2D
3D
TSV
Prolactin receptor
Kd:
2
1
11
2D
3D
TSV
Prolyl oligopeptidase family protein
IC50:
2
1
1
2D
3D
TSV
Prostaglandin G/H synthase 2 [18-504,V335L]
IC50:
2
1
4
2D
3D
TSV
Prostaglandin G/H synthase 2 [18-604,R106Q]
IC50:
2
1
4
2D
3D
TSV
Prostaglandin G/H synthase 2 [18-604,S516A]
IC50:
2
1
4
2D
3D
TSV
Prostaglandin G/H synthase 2 [18-604,V509I]
IC50:
2
1
4
2D
3D
TSV
Prostaglandin G/H synthase 2 [18-604,Y541F]
IC50:
2
1
4
2D
3D
TSV
Proteasome subunit alpha type-2
IC50:
6
1
3
2D
3D
TSV
Protective antigen
EC50:
8
1
7
2D
3D
TSV
Protein kinase C alpha type/glutamine gamma-glutamyltransferase 2
IC50:
2
1
12
2D
3D
TSV
Protein lifeguard 1
Ki:
1
IC50:
1
2
2
2D
3D
TSV
Protein-cysteine N-palmitoyltransferase HHAT
IC50:
2
1
14
2D
3D
TSV
Proto-oncogene Mas
IC50:
2
1
5
2D
3D
TSV
Proto-oncogene tyrosine-protein kinase receptor Ret [638-1114]
IC50:
2
1
6
2D
3D
TSV
Proto-oncogene tyrosine-protein kinase ROS/Sodium-dependent phosphate transport protein 2B
IC50:
2
1
8
2D
3D
TSV
Proto-oncogene tyrosine-protein kinase Src [T341M]
IC50:
2
1
6
2D
3D
TSV
Putative agmatine deiminase
IC50:
2
1
3
2D
3D
TSV
Queuine tRNA-ribosyltransferase catalytic subunit 1
Ki:
2
1
5
2D
3D
TSV
Quinolone signal response protein
Kd:
2
1
3
2D
3D
TSV
RAF proto-oncogene serine/threonine-protein kinase/Serine/threonine-protein kinase B-raf
EC50:
2
1
17
2D
3D
TSV
Replicase polyprotein 1a/Z-RLRGG-AMC
Ki:
2
1
2
2D
3D
TSV
REST corepressor 3
IC50:
2
1
8
2D
3D
TSV
Ret proto-oncogene
Ki:
2
1
1
2D
3D
TSV
Retinoic acid receptor alpha [200-419]/gamma [183-417]
Ki:
2
1
18
2D
3D
TSV
Rho Transcription Termination Factor
ITC:
3
1
5
2D
3D
TSV
Rhodopsin
IC50:
2
EC50:
2
1
1
2D
3D
TSV
Rhomboid protease AarA
IC50:
2
1
1
2D
3D
TSV
Rhomboid protease GluP [F193S,L370F,L379S,R499W]
IC50:
2
1
4
2D
3D
TSV
Rhomboid-related protein 1
IC50:
2
1
1
2D
3D
TSV
Rhomboid-related protein 3
IC50:
2
1
1
2D
3D
TSV
Ribonucleoside-diphosphate reductase large subunit/subunit M2 B
Ki:
1
IC50:
1
2
13
2D
3D
TSV
Ribose-5-phosphate isomerase B
Ki:
3
1
5
2D
3D
TSV
RNA-directed RNA polymerase catalytic subunit
EC50:
3
2
5
2D
3D
TSV
RuvB-like 1
IC50:
2
1
9
2D
3D
TSV
S-adenosylmethionine synthase
IC50:
2
1
1
2D
3D
TSV
Secretin receptor
Ki:
2
EC50:
2
1
5
2D
3D
TSV
Sensor histidine kinase WalK
IC50:
2
1
1
2D
3D
TSV
Serine/threonine-protein kinase CAK1
IC50:
2
1
3
2D
3D
TSV
Serine/threonine-protein kinase KIN28
IC50:
2
1
3
2D
3D
TSV
Serine/threonine-protein kinase N3
IC50:
3
3
3
2D
3D
TSV
Serine/threonine-protein kinase Sgk2 [61-427]
IC50:
2
2
7
2D
3D
TSV
Serine/threonine-protein kinase WNK1 [198-401]
IC50:
4
1
15
2D
3D
TSV
Serine/threonine-protein phosphatase 2B catalytic subunit beta isoform
IC50:
2
2
6
2D
3D
TSV
Short transient receptor potential channel 1/4
IC50:
2
1
14
2D
3D
TSV
Sialyltransferase ST3Gal-I
IC50:
2
1
1
2D
3D
TSV
Signal peptide peptidase-like 2B
IC50:
2
2
10
2D
3D
TSV
Signal transducer and activator of transcription 1-alpha/beta/3
IC50:
2
2
12
2D
3D
TSV
Signal transducer and activator of transcription 4
Kd:
2
2
3
2D
3D
TSV
Small ubiquitin-related modifier 1
IC50:
2
1
8
2D
3D
TSV
Sodium/hydrogen exchanger
IC50:
2
1
1
2D
3D
TSV
Solute carrier family 12 member 2
IC50:
2
1
4
2D
3D
TSV
Solute carrier family 13 member 2
IC50:
3
1
6
2D
3D
TSV
Solute carrier family 13 member 3
IC50:
3
1
17
2D
3D
TSV
Solute carrier organic anion transporter family member 1A2
Ki:
2
1
4
2D
3D
TSV
Spermine oxidase
Ki:
1
IC50:
1
2
18
2D
3D
TSV
Spermine synthase
IC50:
2
1
7
2D
3D
TSV
Spike glycoprotein [668-1255]
EC50:
2
1
8
2D
3D
TSV
Spindlin-2B
Kd:
2
2
3
2D
3D
TSV
Spindlin-3
Kd:
2
2
5
2D
3D
TSV
Spindlin-4
Kd:
2
2
4
2D
3D
TSV
Streptavidin [37-163,Y46S,N47D,S51D,Y107S,R108K,E125D,R127K,E140N]
Kd:
2
1
9
2D
3D
TSV
Stromal interaction molecule 1
IC50:
2
1
4
2D
3D
TSV
Succinate dehydrogenase cytochrome b560 subunit, mitochondrial
Ki:
2
IC50:
1
1
1
2D
3D
TSV
Synaptic vesicular amine transporter [G308A]
IC50:
2
Kd:
1
1
3
2D
3D
TSV
Synaptic vesicular amine transporter [G308P]
IC50:
2
Kd:
1
1
3
2D
3D
TSV
Synaptic vesicular amine transporter [P314G]
IC50:
2
Kd:
1
1
3
2D
3D
TSV
Synaptic vesicular amine transporter [P314L]
IC50:
2
Kd:
1
1
3
2D
3D
TSV
Synaptic vesicular amine transporter [P314T]
IC50:
2
Kd:
1
1
3
2D
3D
TSV
Synaptic vesicular amine transporter [V132A]
IC50:
1
Kd:
1
1
3
2D
3D
TSV
Synaptic vesicular amine transporter [V132G]
IC50:
1
Kd:
1
1
3
2D
3D
TSV
Synaptic vesicular amine transporter [V41A]
IC50:
1
Kd:
1
1
3
2D
3D
TSV
Synaptic vesicular amine transporter [V41I]
IC50:
1
Kd:
1
1
3
2D
3D
TSV
T-cell surface antigen CD2
IC50:
2
1
3
2D
3D
TSV
Testis-specific serine/threonine-protein kinase 6
IC50:
3
3
5
2D
3D
TSV
Topoisomerase I
IC50:
2
1
1
2D
3D
TSV
Trans-sialidase [3-643,Y342H]
Kd:
2
1
2
2D
3D
TSV
Trans-sialidase [3-643]
Kd:
2
1
1
2D
3D
TSV
Transcription factor NF-E2 45 kDa subunit
IC50:
2
1
4
2D
3D
TSV
Transcription factor Sp1
IC50:
2
1
9
2D
3D
TSV
Transcriptional enhancer factor TEF-4
IC50:
2
2
6
2D
3D
TSV
Transcriptional enhancer factor TEF-5
IC50:
2
2
5
2D
3D
TSV
Transcriptional Regulator TtgR Mutant R176G
ITC:
2
1
1
2D
3D
TSV
Transducer protein HtrVI
Ki:
2
2
1
2D
3D
TSV
Transient receptor potential cation channel subfamily M member 7
IC50:
2
2
15
2D
3D
TSV
Troponin C, slow skeletal and cardiac muscles [4-85]
Kd:
2
1
5
2D
3D
TSV
Tubulin
ITC:
2
1
3
2D
3D
TSV
Tubulin beta-4B chain
IC50:
2
1
4
2D
3D
TSV
TyR1
EC50:
2
1
1
2D
3D
TSV
Tyrosine-protein kinase BAZ1B
Kd:
2
1
9
2D
3D
TSV
Tyrosine-protein kinase JAK1 [852-1142]
IC50:
2
1
4
2D
3D
TSV
Tyrosine-protein kinase JAK2 [809-1153]
IC50:
2
1
4
2D
3D
TSV
Tyrosine-protein kinase transforming protein Src [144-247,E177Q,S178L,E179A,T180R,T181V,C186A,K201L]
Kd:
2
1
8
2D
3D
TSV
Tyrosine-protein kinase transforming protein Src [144-247,E177R,S178L,E179Q,T180R,T181V,C186A,K201L]
Kd:
2
1
8
2D
3D
TSV
Tyrosine-protein kinase transforming protein Src [144-247,T181V,C186A,K201L]
Kd:
2
1
4
2D
3D
TSV
Tyrosine-protein kinase transforming protein Src [144-247]
Kd:
2
1
1
2D
3D
TSV
Tyrosine-protein phosphatase non-receptor type 1 [1-301]
Ki:
2
Kd:
2
1
5
2D
3D
TSV
Tyrosine-protein phosphatase non-receptor type 1 [L119V]
IC50:
2
1
5
2D
3D
TSV
Tyrosine-protein phosphatase non-receptor type 14
IC50:
3
3
3
2D
3D
TSV
Tyrosine-protein phosphatase non-receptor type 2 [V121L]
IC50:
2
1
7
2D
3D
TSV
Ubl carboxyl-terminal hydrolase 18
IC50:
2
1
5
2D
3D
TSV
UDP-glucuronosyltransferase 2B15
IC50:
2
2
7
2D
3D
TSV
UDP-N-acetylglucosamine 1-carboxyvinyltransferase 1
IC50:
3
2
4
2D
3D
TSV
Ultraspiracle isoform B
Ki:
1
IC50:
1
1
1
2D
3D
TSV
Uncharacterized protein [173-650]
IC50:
2
2
1
2D
3D
TSV
Unconventional myosin-Va
IC50:
2
2
4
2D
3D
TSV
Undecaprenyl-diphosphatase
IC50:
2
1
5
2D
3D
TSV
Vancomycin/teicoplanin A-type resistance protein VanA
IC50:
2
1
1
2D
3D
TSV
Xanthine-guanine phosphoribosyltransferase
Ki:
2
1
3
2D
3D
TSV
Zinc finger protein 664
Ki:
2
1
1
2D
3D
TSV