PMID

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Article Title

Organization

Species-dependent uptake of glycylsarcosine but not oseltamivir in Pichia pastoris expressing the rat, mouse, and human intestinal peptide transporter PEPT1.

University Of Michigan

Identification of diarylsulfonamides as agonists of the free fatty acid receptor 4 (FFA4/GPR120).

Glaxosmithkline

Interaction of 31 beta-lactam antibiotics with the H+/peptide symporter PEPT2: analysis of affinity constants and comparison with PEPT1.

Biozentrum Of The Martin-Luther-University Halle-Wittenberg

Interactions of a nonpeptidic drug, valacyclovir, with the human intestinal peptide transporter (hPEPT1) expressed in a mammalian cell line.

Rutgers University

Prodrugs of purine and pyrimidine analogues for the intestinal di/tri-peptide transporter PepT1: affinity for hPepT1 in Caco-2 cells, drug release in aqueous media and in vitro metabolism.

The Royal Danish School Of Pharmacy

The tandem chain extension aldol reaction used for synthesis of ketomethylene tripeptidomimetics targeting hPEPT1.

Biogen Idec

CHO/hPEPT1 cells overexpressing the human peptide transporter (hPEPT1) as an alternative in vitro model for peptidomimetic drugs.

The University Of Michigan

5'-Amino acid esters of antiviral nucleosides, acyclovir, and AZT are absorbed by the intestinal PEPT1 peptide transporter.

University Of Michigan

Proton/peptide cotransporter (PEPT 2) from human kidney: functional characterization and chromosomal localization.

Medical College Of Georgia

Direct evidence for peptide transporter (PepT1)-mediated uptake of a nonpeptide prodrug, valacyclovir.

State University Of New Jersey

Human PEPT1 pharmacophore distinguishes between dipeptide transport and binding.

Pharmaceutical Research Institute

Amino acid ester prodrugs of the antiviral agent 2-bromo-5,6-dichloro-1-(beta-D-ribofuranosyl)benzimidazole as potential substrates of hPEPT1 transporter.

University Of Michigan

Three-dimensional quantitative structure-activity relationship analyses of beta-lactam antibiotics and tripeptides as substrates of the mammalian H+/peptide cotransporter PEPT1.

Martin-Luther-University Halle-Wittenberg

Three-dimensional quantitative structure-activity relationship analyses of peptide substrates of the mammalian H+/peptide cotransporter PEPT1.

Martin-Luther-University Halle-Wittenberg

In vitro characterization of human peptide transporter hPEPT1 interactions and passive permeation studies of short cationic antimicrobial peptides.

University Of Troms£

Enhancing the intestinal absorption of molecules containing the polar guanidino functionality: a double-targeted prodrug approach.

University Of Michigan

Structural requirements for the substrates of the H+/peptide cotransporter PEPT2 determined by three-dimensional quantitative structure-activity relationship analysis.

Martin-Luther-University Halle-Wittenberg

Dipeptidomimetic ketomethylene isosteres as pro-moieties for drug transport via the human intestinal di-/tripeptide transporter hPEPT1: design, synthesis, stability, and biological investigations.

University Of Tromsø

Phe-Gly dipeptidomimetics designed for the di-/tripeptide transporters PEPT1 and PEPT2: synthesis and biological investigations.

University Of Tromsø

Bioactivatable Pseudotripeptidization of Cyclic Dipeptides To Increase the Affinity toward Oligopeptide Transporter 1 for Enhanced Oral Absorption: An Application to Cyclo(l-Hyp-l-Ser) (JBP485).

Dalian Medical University

Differential recognition of beta -lactam antibiotics by intestinal and renal peptide transporters, PEPT 1 and PEPT 2.

Medical College Of Georgia

Interaction of anionic cephalosporins with the intestinal and renal peptide transporters PEPT 1 and PEPT 2.

Medical College Of Georgia

Valacyclovir: a substrate for the intestinal and renal peptide transporters PEPT1 and PEPT2.

Medical College Of Georgia

Evidence for the absolute conformational specificity of the intestinal H+/peptide symporter, PEPT1.

Martin-Luther-University Halle-Wittenberg

Human dipeptide transporter, hPEPT1, stably transfected into Chinese hamster ovary cells.

University Of California San Francisco

A novel inhibitor of the mammalian peptide transporter PEPT1.

Martin-Luther-University Halle-Wittenberg

Transport characteristics of differently charged cephalosporin antibiotics in oocytes expressing the cloned intestinal peptide transporter PepT1 and in human intestinal Caco-2 cells.

University Of Giessen