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36 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
28174065 7 Synthesis of new derivatives of 21-imidazolyl-16-dehydropregnenolone as inhibitors of 5a-reductase 2 and with cytotoxic activity in cancer cells.EBI Universidad Nacional Aut£noma de M£xico
27994731 3 Identification of Triptophenolide fromEBI Chinese Academy of Medical Science
23403082 28 Cinnamides as selective small-molecule inhibitors of a cellular model of breast cancer stem cells.EBI Broad Institute of MIT and Harvard
23466225 2 Discovery of AZD3514, a small-molecule androgen receptor downregulator for treatment of advanced prostate cancer.EBI AstraZeneca
16134935 119 Impact of induced fit on ligand binding to the androgen receptor: a multidimensional QSAR study to predict endocrine-disrupting effects of environmental chemicals.EBI University of Basel
17606915 4 Discovery of antiandrogen activity of nonsteroidal scaffolds of marketed drugs.EBI The Scripps Research Institute
16942875 32 A bioisosteric approach to the discovery of indole carbinol androgen receptor ligands.EBI Johnson and Johnson Pharmaceutical Research and Development LLC
16603353 26 Discovery of indole-containing tetracycles as a new scaffold for androgen receptor ligands.EBI Johnson & Johnson Pharmaceutical Research and Development LLC
15454212 16 Synthesis and structure-activity investigation of iodinated arylhydantoins and arylthiohydantoins for development as androgen receptor radioligands.EBI The University of Michigan Medical School
11101354 18 Chiral derivatives of 2-cyclohexylideneperhydro-4,7-methanoindenes, a novel class of nonsteroidal androgen receptor ligand: synthesis, X-ray analysis, and biological activity.EBI The University of Sydney
10966753 5 Design, synthesis, and pharmacological characterization of 4-[4, 4-dimethyl-3-(4-hydroxybutyl)-5-oxo-2-thioxo-1-imidazolidinyl]- 2-iodobenzonitrile as a high-affinity nonsteroidal androgen receptor ligand.EBI The University of Michigan Medical School
1588549 9 Antiandrogenic steroidal sulfonyl heterocycles. Utility of electrostatic complementarity in defining bioisosteric sulfonyl heterocycles.EBI Sterling Winthrop Pharmaceuticals Research Division
3783591 225 Azasteroids: structure-activity relationships for inhibition of 5 alpha-reductase and of androgen receptor binding.EBI TBA
11327585 15 Synthesis and structure-activity studies of side-chain derivatized arylhydantoins for investigation as androgen receptor radioligands.EBI The University of Michigan Medical School
21944856 51 Tetrahydroquinolines as a novel series of nonsteroidal selective androgen receptor modulators: structural requirements for better physicochemical and biological properties.EBI Kaken Pharmaceutical Co., Ltd
21349712 15 Design and synthesis of tricyclic tetrahydroquinolines as a new series of nonsteroidal selective androgen receptor modulators (SARMs).EBI Kaken Pharmaceutical Co., Ltd
17328524 1 Synthesis and biological evaluation of [18F]bicalutamide, 4-[76Br]bromobicalutamide, and 4-[76Br]bromo-thiobicalutamide as non-steroidal androgens for prostate cancer imaging.EBI University of Illinois
17149866 4 Identification of the brominated flame retardant 1,2-dibromo-4-(1,2-dibromoethyl)cyclohexane as an androgen agonist.EBI Orebro University
27131065 26 Design and synthesis of novel bicalutamide and enzalutamide derivatives as antiproliferative agents for the treatment of prostate cancer.EBI School of Pharmacy and Pharmaceutical Sciences
31493989 14 Synthesis, biological evaluation and molecular docking of 4-Amino-2H-benzo[h]chromen-2-one (ABO) analogs containing the piperazine moiety.EBI Luoyang Normal University
31288149 8 A new series of bicalutamide, enzalutamide and enobosarm derivatives carrying pentafluorosulfanyl (SFEBI Cardiff University
30482547 6 Synthesis and biological evaluation of arylpiperazine derivatives as potential anti-prostate cancer agents.EBI Southern Medical University
15715462 70 Three-dimensional structure-activity relationships of nonsteroidal ligands in complex with androgen receptor ligand-binding domain.EBI CSC-Scientific Computing Ltd.
30193215 20 Small molecule-induced degradation of the full length and V7 truncated variant forms of human androgen receptor.EBI Vancouver Prostate Centre (VPC)
28757062 6 Design, synthesis and biological evaluation of novel 3-oxo-4-oxa-5?-androst-17?-amide derivatives as dual 5?-reductase inhibitors and androgen receptor antagonists.EBI China Pharmaceutical University
28937774 107 Selective Nonsteroidal Glucocorticoid Receptor Modulators for the Inhaled Treatment of Pulmonary Diseases.EBI AstraZeneca
28314097 8 Fragment-Sized EthR Inhibitors Exhibit Exceptionally Strong Ethionamide Boosting Effect in Whole-Cell Mycobacterium tuberculosis Assays.BDB University of Cambridge
27250740 15 Electrostatic Control of Isoform Selective Inhibitor Binding in Nitric Oxide Synthase.BDB University of California Irvine
6135157 11 Specific binding of 3H-tiotidine to histamine H2 receptors in guinea pig cerebral cortex.BDB Hoechst Pharmaceutical Research Laboratories
10908357 9 Recognition of a cognate RNA aptamer by neomycin B: quantitative evaluation of hydrogen bonding and electrostatic interactions.BDB The Ohio State University