Search by Compound Name
Compounds Sorted by Binding Targets per Compound
1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 2930 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55
56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 73 74 75 76 77 79 81 84 86 89 95
96 100 108 109 120 124 130 137 143 154 156 168 186 224 240 259 276 278 284 303
304 310 315 323 339 369 370 371 372 373 374 375 376 377 378 380 381 383 384
385 386 388 389 390 391 392 393 394 395 397 398 401 403 404 406 408 418 427
429 443 447 515
Compounds Sorted Alphabetically
Compound Name (alphabetical)
Binding Targets
Enz. Inhib. Data
ITC Data
Alternate Compound Names
- ALK tyrosine kinase receptor
- Activin receptor type-1B
- Angiopoietin-1 receptor
- Apoptosis Signal-regulating Kinase 1 (ASK1)
- Aurora kinase A/Targeting protein for Xklp2
- Axin-1/Glycogen synthase kinase-3 beta
- BDNF/NT-3 growth factors receptor
- BR serine/threonine-protein kinase 1
- CAMK2B
- CDK2/CycE
- CDK2/Cyclin A/Cyclin A1
- Calcium/calmodulin-dependent protein kinase type II subunit delta
- Casein kinase I isoform alpha
- Casein kinase II subunit alpha
- Cyclin-Dependent Kinase 1 (CDK1)
- Cyclin-Dependent Kinase 5 (CDK5)
- Cyclin-Dependent Kinase 9 (CDK9)
- Cytochrome P450 3A
- Cytoplasmic tyrosine-protein kinase BMX
- Death-associated protein kinase 1
- Death-associated protein kinase 3
- Discoidin domain-containing receptor 2
- EPHB1
- Ephrin receptor
- Ephrin type-A receptor 1 (EPHA1)
- Ephrin type-A receptor 2
- Ephrin type-A receptor 3 (EPHA3)
- Ephrin type-B receptor 2
- Ephrin type-B receptor 3 (EPHB3)
- Ephrin type-B receptor 4
- Epidermal growth factor receptor
- Fibroblast growth factor receptor 1
- Fibroblast growth factor receptor 2
- Fibroblast growth factor receptor 3
- Fibroblast growth factor receptor 4
- Focal adhesion kinase 1
- G protein-coupled receptor kinase 5
- G protein-coupled receptor kinase 6
- Hepatocyte growth factor receptor
- High affinity nerve growth factor receptor
- Homeodomain-interacting protein kinase 1
- Homeodomain-interacting protein kinase 3
- Inhibitor of nuclear factor kappa-B kinase subunit beta
- Insulin receptor
- Insulin receptor-related protein
- Insulin-like growth factor I receptor
- Interleukin-1 receptor-associated kinase 1
- Interleukin-1 receptor-associated kinase 4
- MAP kinase p38
- MAP kinase-activated protein kinase 2
- MAP kinase-activated protein kinase 3
- MAP kinase-activated protein kinase 5
- MAP/microtubule affinity-regulating kinase 2
- Macrophage colony-stimulating factor 1 receptor (CSF1R)
- Macrophage-stimulating protein receptor
- Misshapen-like kinase 1
- Mitogen-activated protein kinase 1
- Mitogen-activated protein kinase 10
- Mitogen-activated protein kinase 11
- Mitogen-activated protein kinase 12
- Mitogen-activated protein kinase 13 (MAPK13)
- Mitogen-activated protein kinase 14
- Mitogen-activated protein kinase 3
- Mitogen-activated protein kinase 8
- Mitogen-activated protein kinase 9
- Mitogen-activated protein kinase kinase kinase 9 (MLK1)
- NUAK family SNF1-like kinase 1
- PAS domain-containing serine/threonine-protein kinase
- PKC alpha and beta-2
- PTK2B protein tyrosine kinase 2 beta (PTK2B)
- Phosphorylase kinase
- Platelet-derived growth factor receptor alpha
- Platelet-derived growth factor receptor beta
- Polycystin-2
- Protein kinase C alpha type
- Protein kinase C delta type
- Protein kinase C theta type
- Protein kinase C, eta
- Protein kinase C, gamma
- Proto-oncogene tyrosine-protein kinase ROS
- Proto-oncogene tyrosine-protein kinase Src
- Proto-oncogene tyrosine-protein kinase receptor Ret
- RAC-alpha serine/threonine-protein kinase
- Receptor protein-tyrosine kinase erbB-4
- Rho-associated protein kinase 1
- Rho-associated protein kinase 2
- Ribosomal protein S6 kinase (P70S6K)
- Ribosomal protein S6 kinase alpha 1
- Ribosomal protein S6 kinase alpha 4
- Ribosomal protein S6 kinase alpha 5
- Serine/threonine protein kinase NLK
- Serine/threonine-protein kinase 17A
- Serine/threonine-protein kinase 33
- Serine/threonine-protein kinase 4 (STK4)
- Serine/threonine-protein kinase AKT
- Serine/threonine-protein kinase AKT2
- Serine/threonine-protein kinase CHK2
- Serine/threonine-protein kinase Chk1/2
- Serine/threonine-protein kinase D1
- Serine/threonine-protein kinase MARK1
- Serine/threonine-protein kinase MST2
- Serine/threonine-protein kinase Nek3
- Serine/threonine-protein kinase PAK 4
- Serine/threonine-protein kinase PAK6
- Serine/threonine-protein kinase PAK7
- Serine/threonine-protein kinase PLK1
- Serine/threonine-protein kinase PLK2
- Serine/threonine-protein kinase PLK3
- Serine/threonine-protein kinase PRKX
- Serine/threonine-protein kinase RIPK2
- Serine/threonine-protein kinase Sgk1
- Serine/threonine-protein kinase TBK1
- Serine/threonine-protein kinase WNK2
- Serine/threonine-protein kinase pim-1
- Serine/threonine-protein kinase pim-2
- Testis-specific serine/threonine-protein kinase 2
- Tyrosine-protein kinase ABL1
- Tyrosine-protein kinase ABL2
- Tyrosine-protein kinase BRK
- Tyrosine-protein kinase BTK
- Tyrosine-protein kinase Blk
- Tyrosine-protein kinase CSK
- Tyrosine-protein kinase FER
- Tyrosine-protein kinase Fes/Fps
- Tyrosine-protein kinase Fgr
- Tyrosine-protein kinase Fyn
- Tyrosine-protein kinase HCK
- Tyrosine-protein kinase JAK2
- Tyrosine-protein kinase JAK3
- Tyrosine-protein kinase Lck
- Tyrosine-protein kinase Lyn
- Tyrosine-protein kinase SYK
- Tyrosine-protein kinase Yes
- Tyrosine-protein kinase ZAP-70
- Tyrosine-protein kinase receptor FLT3
- Tyrosine-protein kinase receptor UFO
- Vascular endothelial growth factor receptor 1
- Vascular endothelial growth factor receptor 2
- Vascular endothelial growth factor receptor 3
- [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial
- cGMP-dependent protein kinase
- p21-Activated kinase 2 (PAK2)
- p21-Activated kinase 3 (PAK3)
148 IC50
- CHEMBL1929238