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Compounds Sorted by Binding Targets per Compound

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Compounds Sorted Alphabetically
Compound Name (alphabetical)
Binding Targets
Enz. Inhib. Data
ITC Data
Alternate Compound Names
  • ALK tyrosine kinase receptor
  • Activin receptor type-1B
  • Angiopoietin-1 receptor
  • Apoptosis Signal-regulating Kinase 1 (ASK1)
  • Aurora kinase A/Targeting protein for Xklp2
  • Axin-1/Glycogen synthase kinase-3 beta
  • BDNF/NT-3 growth factors receptor
  • BR serine/threonine-protein kinase 1
  • CAMK2B
  • CDK2/CycE
  • CDK2/Cyclin A/Cyclin A1
  • Calcium/calmodulin-dependent protein kinase type II subunit delta
  • Casein kinase I isoform alpha
  • Casein kinase II subunit alpha
  • Cyclin-Dependent Kinase 1 (CDK1)
  • Cyclin-Dependent Kinase 5 (CDK5)
  • Cyclin-Dependent Kinase 9 (CDK9)
  • Cytochrome P450 3A
  • Cytoplasmic tyrosine-protein kinase BMX
  • Death-associated protein kinase 1
  • Death-associated protein kinase 3
  • Discoidin domain-containing receptor 2
  • EPHB1
  • Ephrin receptor
  • Ephrin type-A receptor 1 (EPHA1)
  • Ephrin type-A receptor 2
  • Ephrin type-A receptor 3 (EPHA3)
  • Ephrin type-B receptor 2
  • Ephrin type-B receptor 3 (EPHB3)
  • Ephrin type-B receptor 4
  • Epidermal growth factor receptor
  • Fibroblast growth factor receptor 1
  • Fibroblast growth factor receptor 2
  • Fibroblast growth factor receptor 3
  • Fibroblast growth factor receptor 4
  • Focal adhesion kinase 1
  • G protein-coupled receptor kinase 5
  • G protein-coupled receptor kinase 6
  • Hepatocyte growth factor receptor
  • High affinity nerve growth factor receptor
  • Homeodomain-interacting protein kinase 1
  • Homeodomain-interacting protein kinase 3
  • Inhibitor of nuclear factor kappa-B kinase subunit beta
  • Insulin receptor
  • Insulin receptor-related protein
  • Insulin-like growth factor I receptor
  • Interleukin-1 receptor-associated kinase 1
  • Interleukin-1 receptor-associated kinase 4
  • MAP kinase p38
  • MAP kinase-activated protein kinase 2
  • MAP kinase-activated protein kinase 3
  • MAP kinase-activated protein kinase 5
  • MAP/microtubule affinity-regulating kinase 2
  • Macrophage colony-stimulating factor 1 receptor (CSF1R)
  • Macrophage-stimulating protein receptor
  • Misshapen-like kinase 1
  • Mitogen-activated protein kinase 1
  • Mitogen-activated protein kinase 10
  • Mitogen-activated protein kinase 11
  • Mitogen-activated protein kinase 12
  • Mitogen-activated protein kinase 13 (MAPK13)
  • Mitogen-activated protein kinase 14
  • Mitogen-activated protein kinase 3
  • Mitogen-activated protein kinase 8
  • Mitogen-activated protein kinase 9
  • Mitogen-activated protein kinase kinase kinase 9 (MLK1)
  • NUAK family SNF1-like kinase 1
  • PAS domain-containing serine/threonine-protein kinase
  • PKC alpha and beta-2
  • PTK2B protein tyrosine kinase 2 beta (PTK2B)
  • Phosphorylase kinase
  • Platelet-derived growth factor receptor alpha
  • Platelet-derived growth factor receptor beta
  • Polycystin-2
  • Protein kinase C alpha type
  • Protein kinase C delta type
  • Protein kinase C theta type
  • Protein kinase C, eta
  • Protein kinase C, gamma
  • Proto-oncogene tyrosine-protein kinase ROS
  • Proto-oncogene tyrosine-protein kinase Src
  • Proto-oncogene tyrosine-protein kinase receptor Ret
  • RAC-alpha serine/threonine-protein kinase
  • Receptor protein-tyrosine kinase erbB-4
  • Rho-associated protein kinase 1
  • Rho-associated protein kinase 2
  • Ribosomal protein S6 kinase (P70S6K)
  • Ribosomal protein S6 kinase alpha 1
  • Ribosomal protein S6 kinase alpha 4
  • Ribosomal protein S6 kinase alpha 5
  • Serine/threonine protein kinase NLK
  • Serine/threonine-protein kinase 17A
  • Serine/threonine-protein kinase 33
  • Serine/threonine-protein kinase 4 (STK4)
  • Serine/threonine-protein kinase AKT
  • Serine/threonine-protein kinase AKT2
  • Serine/threonine-protein kinase CHK2
  • Serine/threonine-protein kinase Chk1/2
  • Serine/threonine-protein kinase D1
  • Serine/threonine-protein kinase MARK1
  • Serine/threonine-protein kinase MST2
  • Serine/threonine-protein kinase Nek3
  • Serine/threonine-protein kinase PAK 4
  • Serine/threonine-protein kinase PAK6
  • Serine/threonine-protein kinase PAK7
  • Serine/threonine-protein kinase PLK1
  • Serine/threonine-protein kinase PLK2
  • Serine/threonine-protein kinase PLK3
  • Serine/threonine-protein kinase PRKX
  • Serine/threonine-protein kinase RIPK2
  • Serine/threonine-protein kinase Sgk1
  • Serine/threonine-protein kinase TBK1
  • Serine/threonine-protein kinase WNK2
  • Serine/threonine-protein kinase pim-1
  • Serine/threonine-protein kinase pim-2
  • Testis-specific serine/threonine-protein kinase 2
  • Tyrosine-protein kinase ABL1
  • Tyrosine-protein kinase ABL2
  • Tyrosine-protein kinase BRK
  • Tyrosine-protein kinase BTK
  • Tyrosine-protein kinase Blk
  • Tyrosine-protein kinase CSK
  • Tyrosine-protein kinase FER
  • Tyrosine-protein kinase Fes/Fps
  • Tyrosine-protein kinase Fgr
  • Tyrosine-protein kinase Fyn
  • Tyrosine-protein kinase HCK
  • Tyrosine-protein kinase JAK2
  • Tyrosine-protein kinase JAK3
  • Tyrosine-protein kinase Lck
  • Tyrosine-protein kinase Lyn
  • Tyrosine-protein kinase SYK
  • Tyrosine-protein kinase Yes
  • Tyrosine-protein kinase ZAP-70
  • Tyrosine-protein kinase receptor FLT3
  • Tyrosine-protein kinase receptor UFO
  • Vascular endothelial growth factor receptor 1
  • Vascular endothelial growth factor receptor 2
  • Vascular endothelial growth factor receptor 3
  • [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial
  • cGMP-dependent protein kinase
  • p21-Activated kinase 2 (PAK2)
  • p21-Activated kinase 3 (PAK3)
148 IC50
  • CHEMBL1929238