Search by Compound Name
Compounds Sorted by Binding Targets per Compound
1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 2930 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55
56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 73 74 75 76 77 79 81 84 86 89 95
96 100 108 109 120 124 130 137 143 154 156 168 186 224 240 259 276 278 284 303
304 310 315 323 339 369 370 371 372 373 374 375 376 377 378 380 381 383 384
385 386 388 389 390 391 392 393 394 395 397 398 401 403 404 406 408 418 427
429 443 447 515
Compounds Sorted Alphabetically
Compound Name (alphabetical)
Binding Targets
Enz. Inhib. Data
ITC Data
Alternate Compound Names
- Bile salt export pump
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- GABA A Alpha2Beta1Gamma2
- GABA A Alpha4Beta2Gamma2
- GABA A receptor alpha-2/beta-2/gamma-2
- GABA A receptor alpha-3/beta-2/gamma-2
- GABA A receptor alpha-5/beta-3/gamma-2
- GABA A receptor alpha-6/beta-2/gamma-2
- GABA receptor alpha-1/beta-2/gamma-2 subunit
- GABA receptor alpha-1/beta-3/gamma-2 subunit
- GABA receptor alpha-2/beta-2/gamma-2 subunit
- GABA receptor alpha-2/beta-3/gamma-2 subunit
- GABA receptor alpha-3/beta-2/gamma-2 subunit
- GABA receptor alpha-3/beta-3/gamma-2 subunit
- GABA receptor alpha-5/beta-3/gamma-2 subunit
- GABA receptor alpha-6/beta-2/gamma-2 subunit
- GABA receptor alpha-6/beta-3/gamma-2 subunit
- GABA(A) receptor subunit alpha-2
- GABA-A receptor; alpha-1/beta-2/gamma-2
- GABAA Receptor Mutant, alpha-1 (A160C), beta-2, gamma-2
- GABAA Receptor Mutant, alpha-1 (F99C), beta-2, gamma-2
- GABAA Receptor Mutant, alpha-1 (G157C), beta-2, gamma-2
- GABAA Receptor Mutant, alpha-1 (G200C), beta-2, gamma-2
- GABAA Receptor Mutant, alpha-1 (S204C), beta-2, gamma-2
- GABAA Receptor Mutant, alpha-1 (S205C), beta-2, gamma-2
- GABAA Receptor Mutant, alpha-1 (T162C), beta-2, gamma-2
- GABAA Receptor Mutant, alpha-1 (T206C), beta-2, gamma-2
- GABAA Receptor Mutant, alpha-1 (V202C), beta-2, gamma-2
- GABAA Receptor Mutant, alpha-1 (V211C), beta-2, gamma-2
- GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (A79C)
- GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (Chimera)
- GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (D56C)
- GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (L140C)
- GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (M130C)
- GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (R132C)
- GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (R144C)
- GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (R185C)
- GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (R194C)
- GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (T126C)
- GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (T142C)
- GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (T81C)
- GABAA Receptor, alpha-1, beta-2, gamma-2
- GABAA Receptor, alpha-2, beta-2, gamma-2
- GABAA Receptor, alpha-3, beta-2, gamma-2
- GABAA Receptor, alpha-4, beta-2, gamma-2
- GABAA Receptor, alpha-5, beta-2, gamma-2
- GABAA Receptor, alpha-6, beta-2, gamma-2
- Gamma-aminobutyric acid receptor subunit alpha-1
- Gamma-aminobutyric acid receptor subunit alpha-3
- Gamma-aminobutyric acid receptor subunit alpha-5 (GABA(A))
- Gamma-aminobutyric acid type B receptor subunit 1
- Multidrug resistance-associated protein 4
- Peripheral-Type Benzodiazepine Receptor
- Serum albumin
- Ambien
- CHEMBL911
- Dalparan
- N,N-dimethyl-2-[6-methyl-2-(4-methylphenyl)imidazo[1,2-a]pyridin-3-yl]acetamide
- ZPM
- Zolpidem
- Zolpidem tartrate
- 1,3-beta-glucan synthase component GLS2
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2B
- 5-hydroxytryptamine receptor 2C
- Acetylcholinesterase
- Adrenergic receptor alpha-2
- Alpha-1 Adrenergic Receptor/ adrenergic receptor/ adrenergic receptor
- Alpha-1A adrenergic receptor
- Alpha-2A adrenergic receptor
- Beta-2 adrenergic receptor
- Bile salt export pump
- Calcium channel
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- Cytochrome P450
- Cytochrome P450 1B1
- Cytochrome P450 2C19
- Cytochrome P450 2C8
- Cytochrome P450 2J2
- D(1A) dopamine receptor
- D(2) dopamine receptor
- Dopamine transporter
- HTR1D
- HTR2C
- HTR6
- Histamine H1 receptor
- Histamine H3 receptor
- Monoamine transporters; Norepininephrine & dopamine
- Multidrug resistance protein 1/Multidrug resistance associated protein 1
- Multidrug resistance-associated protein 4
- Muscarinic acetylcholine receptor M1
- Muscarinic acetylcholine receptor M2
- Muscarinic acetylcholine receptor M3
- Muscarinic acetylcholine receptor M4
- Muscarinic acetylcholine receptor M5
- Norepinephrine Monoamine transporters
- Norepinephrine transporter
- Potassium voltage-gated channel subfamily C member 1
- Potassium voltage-gated channel subfamily H member 2
- SLC6A3
- Serotonin (5-HT) receptor
- Serotonin 1 (5-HT1) receptor
- Serotonin 1B/1D receptor
- Serotonin 2 (5-HT2) receptor
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- Serum albumin
- Sigma non-opioid intracellular receptor 1
- Sodium-dependent dopamine transporter
- Sodium-dependent noradrenaline transporter
- Sodium-dependent serotonin transporter
- Transporter
- Twik-RElated Potassium (K+) channel 1 (TREK1)
- adrenergic Alpha2
- ubiquitin-conjugating enzyme E2 N
- CHEMBL1201082
- CHEMBL41
- Fluoxetin
- Fluoxetine
- Prozac
- US9120771, Fluoxetine
- cid_62857
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 1D
- 5-hydroxytryptamine receptor 3A
- 5-hydroxytryptamine receptor 5A
- 5-hydroxytryptamine receptor 6
- 5-hydroxytryptamine receptor 7
- Acetylcholinesterase
- Adrenergic alpha1B
- Aldose reductase
- Alpha-1A adrenergic receptor
- Alpha-2A adrenergic receptor
- Alpha-2B adrenergic receptor
- Alpha-2C adrenergic receptor
- Alpha-chymotrypsin
- Axin-1/Glycogen synthase kinase-3 beta
- Beta-1 adrenergic receptor
- Beta-2 adrenergic receptor
- Beta-lactamase
- Cholinesterases
- Cytochrome P450 3A
- D(1A) dopamine receptor
- D(1B) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- Dihydroorotate dehydrogenase (fumarate)
- Dopamine receptor
- EBifunctional epoxide hydrolase 2
- Gamma-aminobutyric acid receptor subunit alpha-1
- Genome polyprotein
- Glutamate receptor ionotropic, NMDA 1
- Histamine H1 receptor
- Kappa-type opioid receptor
- L-lactate dehydrogenase A chain
- Lysine-specific histone demethylase 1A
- Mitogen-activated protein kinase 14
- Mu-type opioid receptor
- Muscarinic acetylcholine receptor M1
- Muscarinic acetylcholine receptor M2
- Muscarinic acetylcholine receptor M3
- Muscarinic acetylcholine receptor M4
- Muscarinic acetylcholine receptor M5
- Neuraminidase
- Neuromedin-U receptor 2
- OPRD1
- SLC6A3
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- Serum albumin
- Sialidase
- Sodium-dependent noradrenaline transporter
- Sodium-dependent serotonin transporter
- Trypsin
- Tyrosinase
- Vasopressin V1b receptor
- Vasopressin V2 receptor
- Xanthine dehydrogenase/oxidase
- 2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4H-chromen-3-yl 6-O-(6-deoxy-alpha-L-mannopyranosyl)-beta-D-glucopyranoside
- 3-Rhamnoglucosylquercetin
- 3-Rutinosyl quercetin
- CHEMBL226335
- cid_5280805
- rutin
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 1B
- 5-hydroxytryptamine receptor 1D
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 3A
- 5-hydroxytryptamine receptor 5A
- 5-hydroxytryptamine receptor 6
- 5-hydroxytryptamine receptor 7
- Adrenergic alpha1B
- Alpha-1A adrenergic receptor
- Alpha-2A adrenergic receptor
- Alpha-2B adrenergic receptor
- Alpha-2C adrenergic receptor
- Beta-1 adrenergic receptor
- Beta-2 adrenergic receptor
- Calcium channel
- Cannabinoid receptor 1
- Cholinergic, Nicotinic Alpha3Beta2
- Cystine/glutamate transporter
- D(1A) dopamine receptor
- D(1B) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- Dopamine receptor
- Gamma-aminobutyric acid receptor subunit alpha-1
- Glutamate receptor ionotropic, NMDA 1
- Histamine H1 receptor
- Histamine H2 Receptor
- Histamine H4 receptor
- Imidazoline I1
- Kappa-type opioid receptor
- Metabotropic glutamate receptor
- Metabotropic glutamate receptor 1
- Metabotropic glutamate receptor 2
- Metabotropic glutamate receptor 4 (mGlu4)
- Metabotropic glutamate receptor 4 (mGluR4)
- Metabotropic glutamate receptor 5
- Metabotropic glutamate receptor 6 (mGlu6)
- Metabotropic glutamate receptor 8 (mGlu8)
- Mu-type opioid receptor
- Muscarinic acetylcholine receptor M1
- Muscarinic acetylcholine receptor M2
- Muscarinic acetylcholine receptor M3
- Muscarinic acetylcholine receptor M4
- Muscarinic acetylcholine receptor M5
- Neuronal acetylcholine receptor
- Neuronal acetylcholine receptor subunit alpha-4
- Neuronal acetylcholine receptor; alpha2/beta2
- Oxytocin receptor
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- Sodium-dependent dopamine transporter
- Sodium-dependent noradrenaline transporter
- Sodium-dependent serotonin transporter
- Vasopressin V1b receptor
- Vasopressin V2 receptor
- (S)-2-amino-4-sulfobutanoic acid
- CHEMBL230951
- L-2-amino-4-sulfobutyric acid
- L-Homocysteate
- L-homocysteic acid