Search by Compound Name
Compounds Sorted by Binding Targets per Compound
1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 2930 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55
56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 73 74 75 76 77 79 81 84 86 89 95
96 100 108 109 120 124 130 137 143 154 156 168 186 224 240 259 276 278 284 303
304 310 315 323 339 369 370 371 372 373 374 375 376 377 378 380 381 383 384
385 386 388 389 390 391 392 393 394 395 397 398 401 403 404 406 408 418 427
429 443 447 515
Compounds Sorted Alphabetically
Compound Name (alphabetical)
Binding Targets
Enz. Inhib. Data
ITC Data
Alternate Compound Names
- 5-HT1
- 5-HT3A Serotonin Receptor
- 5-Hydroxytryptamine receptor 6 (5-HT6)
- 5-Hydroxytryptamine receptor 7 (5-HT7)
- 5-hydroxytryptamine receptor 1A (5-HT1A)
- 5-hydroxytryptamine receptor 1B
- 5-hydroxytryptamine receptor 1D
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2C
- 5-hydroxytryptamine receptor 7 (5HT7)
- ADRA1A
- ADRA1B
- ADRA2C
- ADRB2
- Adenosine Receptors A2a (A2a)
- Adenosine receptor A1
- Adrenergic receptor alpha-2
- Alpha adrenergic receptor 1A and 1B
- Alpha-1A adrenergic receptor
- Alpha-2A adrenergic receptor
- Alpha-2B adrenergic receptor
- Alpha-2C adrenergic receptor
- Angiotensin II AT2
- Angiotensin II type 1a (AT-1a) receptor
- Beta-1 adrenergic receptor
- Beta-2 adrenergic receptor and beta-3 adrenergic receptor
- CCKBR
- CHRM5
- Calcium channel
- Cholecystokinin B
- Cholinergic, muscarinic
- Cysteinyl leukotriene receptor 1
- D(1A) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- DOPAMINE
- DRD1
- DRD2
- DRD3
- Delta-type opioid receptor
- Dopamine D1 receptor
- Dopamine D2 receptor
- Dopamine D2 receptor/Serotonin 2 (5-HT2) receptor
- Dopamine D5 receptor
- Dopamine Transporter (DAT)
- Dopamine receptor
- Dopamine receptors; D2 & D4
- GRIA3
- Gamma-aminobutyric acid receptor subunit alpha-1 (GABA(A) alpha-1)
- Gamma-aminobutyric acid type B receptor subunit 1
- Glutamate kainate
- Glycine
- Glycine, non-strychnine
- HRH3
- HTR1D
- HTR2C
- HTR4
- HTR6
- HTR7
- Histamine H1 receptor
- Histamine H4 receptor
- Histamine receptor (H3)
- Imidazoline I1
- Ionotropic glutamate receptor NMDA 1/2D
- Kappa-type opioid receptor
- Muscarinic acetylcholine receptor M1
- Muscarinic acetylcholine receptor M2
- Muscarinic acetylcholine receptor M3
- Muscarinic acetylcholine receptor M4
- NT
- Nociceptin/mu opioid receptor
- Norepinephrine transporter
- Prostanoid TP receptor
- Serotonin (5-HT) receptor
- Serotonin 1B/1D receptor
- Serotonin receptor (2b and 2c)
- Serotonin receptor 2a and 2b (5HT2A and 5HT2B)
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- Sigma non-opioid intracellular receptor 1
- Sodium-dependent serotonin transporter
- Substance P
- Voltage-gated sodium channel subunit alpha Nav1.8
- adrenergic Alpha2
- 6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatricyclo[9.4.0.0^{3,8}]pentadeca-1,3(8),4,6,10,12,14-heptaene
- CLOZARIL
- Clozapine
- Leponex
- 1,3-beta-glucan synthase component GLS2
- 5-HT3A Serotonin Receptor
- 5-Hydroxytryptamine receptor 6 (5-HT6)
- 5-Hydroxytryptamine receptor 7 (5-HT7)
- 5-hydroxytryptamine receptor 1A (5-HT1A)
- 5-hydroxytryptamine receptor 1A (5HT1A)
- 5-hydroxytryptamine receptor 1B
- 5-hydroxytryptamine receptor 1D
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2C
- 5-hydroxytryptamine receptor 7 (5HT7)
- ADRA1A
- ADRA1B
- Adrenergic receptor alpha
- Adrenergic receptor alpha-1
- Adrenergic receptor alpha-2
- Adrenergic receptor beta
- Alpha-1 Adrenergic Receptor/ adrenergic receptor/ adrenergic receptor
- Alpha-1A adrenergic receptor
- Alpha-2A adrenergic receptor
- Alpha-2B adrenergic receptor
- Alpha-2C adrenergic receptor
- Beta-1 adrenergic receptor
- Beta-2 adrenergic receptor and beta-3 adrenergic receptor
- Bile salt export pump
- CCKBR
- CHRM5
- Calcium channel
- Calcium channel (Type L)
- Cholecystokinin B
- Cholinergic, muscarinic
- Cysteinyl leukotriene receptor 1
- D(1A) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- DOPAMINE
- DRD2
- Delta-type opioid receptor
- Dopamine D2 receptor
- Dopamine D2 receptor/Serotonin 2 (5-HT2) receptor
- Dopamine D5 receptor
- Dopamine Transporter (DAT)
- Dopamine receptor
- Dopamine receptors; D2 & D4
- Gamma-aminobutyric acid receptor subunit alpha-1 (GABA(A) alpha-1)
- Glycine receptor subunit alpha-1
- HTR1D
- HTR2C
- HTR6
- HTR7
- Histamine H1 receptor
- Histone H1
- Kappa-type opioid receptor
- Multidrug and toxin extrusion protein 1
- Multidrug and toxin extrusion protein 2
- Muscarinic acetylcholine receptor
- Muscarinic acetylcholine receptor M1
- Muscarinic acetylcholine receptor M2
- Muscarinic acetylcholine receptor M3
- Muscarinic acetylcholine receptor M4
- NT
- Nociceptin/mu opioid receptor
- Norepinephrine Monoamine transporters
- Norepinephrine transporter
- Potassium voltage-gated channel subfamily H member 2
- Prostanoid TP receptor
- Serotonin (5-HT) receptor
- Serotonin 1 (5-HT1) receptor
- Serotonin 1B/1D receptor
- Serotonin 2 (5-HT2) receptor
- Serotonin receptor (2b and 2c)
- Serotonin receptor 2a and 2b (5HT2A and 5HT2B)
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- Serum albumin
- Sigma non-opioid intracellular receptor 1
- Sodium channel protein type 5 subunit alpha
- Sodium-dependent serotonin transporter
- Solute carrier family 22 member 2
- Substance P
- Transporter
- Voltage-dependent L-type calcium channel subunit alpha-1C
- Voltage-gated sodium channel subunit alpha Nav1.8
- adrenergic Alpha2
- (risperidone)3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-ethyl}-2-methyl-6,7,8,9-tetrahydro-pyrido[1,2-a]pyrimidin-4-one
- 1-(2-Allyl-phenoxy)-3-isopropylamino-propan-2-ol
- 2-(2-(4-(benzo[d]isoxazol-3-yl)piperidin-1-yl)ethyl)-7,8,9,9a-tetrahydro-1H-pyrido[1,2-a]pyrimidin-4(6H)-one
- 2-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-ethyl}-6,7,8,8a-tetrahydro-5H-naphthalen-1-one
- 3-(2-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)ethyl)-2-methyl-6,7,8,9-tetrahydropyrido[1,2-a]pyrimidin-4-one
- 3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-ethyl}-2-methyl-6,7,8,9-tetrahydro-pyrido[1,2-a]pyrimidin-4-one
- 3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-ethyl}-2-methyl-6,7,8,9-tetrahydro-pyrido[1,2-a]pyrimidin-4-one (Resperidone)
- 3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-ethyl}-2-methyl-6,7,8,9-tetrahydro-pyrido[1,2-a]pyrimidin-4-one (risperidone)
- 3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-ethyl}-2-methyl-6,7,8,9-tetrahydro-pyrido[1,2-a]pyrimidin-4-one(risperidone)
- 5-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-ethyl]-6-methyl-1,3-dihydro-indol-2-one(Norastemizole)
- CHEMBL85
- R 64 766
- RISPERDAL
- RISPERIDONE
- US10167256, Risperidone
- US10174011, risperidone
- US8802672, Risperidone