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Compound Name:

Compounds Sorted by Binding Targets per Compound

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Compounds Sorted Alphabetically

Compound Name (alphabetical)	Binding Targets	Enz. Inhib. Data							ITC Data	Alternate Compound Names
		Ki	IC50	Kd	EC50	Koff	Kon	Other
BDBM22869	5-HT1 5-HT2 5-HT7L 5-HT7S 5-HT7b 5-hydroxytryptamine receptor 1B (5HT1B) 5-hydroxytryptamine receptor 2C (5HT2c) ADRA1A ADRA1B ADRA2B ADRA2C ADRB2 Adenosine receptors; A1 & A2a Adenosine receptors; A1 & A3 Adrenergic receptor alpha Adrenergic receptor beta; ADRB1 & ADRB3 Adrenergic, alpha-2B-, receptor [Homo sapiens] Alpha-1 Adrenergic Receptor Alpha-1 adrenoreceptor Angiotensin II AT2 Angiotensin II type 1a (AT-1a) receptor Benzodiazepine receptors; peripheral & central CCKBR CHRM5 Calcium channel Cholecystokinin B Cholinergic, muscarinic Cysteinyl leukotriene receptor 1 DOPAMINE D2/D4 DOPAMINE D4.2 DOPAMINE D4.4 DRD1 DRD2 DRD3 DRD4 DRD5 Dopamine D1 receptor Dopamine D2A Dopamine Transporter (DAT) Dopamine receptor Dopamine2-like GABA B GABA uptake GRIA3 Glutamate kainate Glutamate-NMDA-Channel Glutamate-NMDA-Polyamine Glycine Glycine, strychnine HRH3 HTR1D HTR1F HTR2A HTR2B HTR2C HTR3A HTR4 HTR6 HTR7 Histamine H1 receptor Histamine H4 Receptor Imidazoline I1 Muscarinic acetylcholine receptor Muscarinic acetylcholine receptor M4 Muscarinic acetylcholine receptors; M1 & M2 Muscarinic receptor M1 and M2 Muscarinic receptor M2 and M3 NT Nociceptin/mu opioid receptor Norepinephrine transporter OPRD1 Serotonin (5-HT) receptor Serotonin (5-HT3) receptor Serotonin 1 receptors; 5-HT1B & 5-HT1D Serotonin 1a (5-HT1a) receptor/Adrenergic receptor alpha-1 Serotonin Receptor 1E Serotonin Transporter (SERT) Sigma Sigma1-receptor Sodium Channel Substance P TBXA2R adrenergic Alpha1 adrenergic Alpha2 mu/kappa opioid receptor	406	3	0	0	0	0	0	0	6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatricyclo[9.4.0.0^{3,8}]pentadeca-1,3(8),4,6,10,12,14-heptaene CLOZARIL Clozapine Leponex