BDBM50011875 2-Bromo-4-(2-chloro-phenyl)-9-methyl-6H-1-thia-5,7,8,9a-tetraaza-cyclopenta[e]azulene::BROTIZOLAM::CHEMBL32479

SMILES Cc1nnc2CN=C(c3cc(Br)sc3-n12)c1ccccc1Cl

InChI Key InChIKey=UMSGKTJDUHERQW-UHFFFAOYSA-N

Data  2 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50011875   

TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Rhone-Poulenc Sante

Curated by PDSP Ki Database
LigandPNGBDBM50011875(2-Bromo-4-(2-chloro-phenyl)-9-methyl-6H-1-thia-5,7...)
Affinity DataKi:  17.4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Rhone-Poulenc Sante

Curated by PDSP Ki Database
LigandPNGBDBM50011875(2-Bromo-4-(2-chloro-phenyl)-9-methyl-6H-1-thia-5,7...)
Affinity DataKi:  80.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Rhone-Poulenc Sante

Curated by PDSP Ki Database
LigandPNGBDBM50011875(2-Bromo-4-(2-chloro-phenyl)-9-methyl-6H-1-thia-5,7...)
Affinity DataIC50:  300nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed