BDBM101515 US8524699, 26::US8530652, 42::US8530670, 31

SMILES CC1(C)N(Cc2c(Nc3ncnc4sccc34)[nH]nc12)C(=O)N[C@@H]1C[C@H]1c1ccccc1

InChI Key InChIKey=AUEJJEQMGQCKCW-DOTOQJQBSA-N

Data  2 KI  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 101515   

TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Agouron Pharmaceuticals

US Patent
LigandPNGBDBM101515(US8524699, 26 | US8530652, 42 | US8530670, 31)
Affinity DataKi:  16nM EC50:  340nMAssay Description:The enzymatic activity of PAK4 KD was measured by its ability to catalyzed the transfer of a phosphate residue from a nucleoside triphosphate to an a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Agouron Pharmaceuticals

US Patent
LigandPNGBDBM101515(US8524699, 26 | US8530652, 42 | US8530670, 31)
Affinity DataKi:  94nM EC50:  610nMAssay Description:The enzymatic activity of PAK4 KD was measured by its ability to catalyzed the transfer of a phosphate residue from a nucleoside triphosphate to an a...More data for this Ligand-Target Pair
In DepthDetails US Patent