BDBM272564 (R)-4-methyl-2-(8-methyl- 5,6,7,8-tetrahydro- [1,2,4]triazolo[4,3-a]pyrazin- 3-yl)oxazole::US10065961, Compound 27::US10941151, Compound 27
SMILES C[C@H]1NCCn2c1nnc2-c1nc(C)co1
InChI Key InChIKey=ZJUWQZAEPLRGCJ-SSDOTTSWSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 272564
Affinity DataKi: 51nMAssay Description:The antagonist activity of compounds of the invention is measured following pre-incubation (3 minutes) of the compound with the cells, followed by ad...More data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:NK3: The ability of compounds of the invention to inhibit the binding of the NK-3 receptor selective antagonist 3H-SB222200 was assessed by an in vit...More data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:The antagonist activity of compounds of the invention is measured following pre-incubation (3 minutes) of the compound with the cells, followed by ad...More data for this Ligand-Target Pair