BDBM296189 2-{4-[(4-isopropyl-phenyl)-(2,2,2-trifluoro- ethyl)-amino]-phenoxy}-pyrido[3,4- d]pyrimidin-4-ol::US10112940, Example 114::US10202381, Example 114::US10208039, Example 114::US10611763, Example 114::US10815234, Example 114::US11535616, Example 114

SMILES CC(C)c1ccc(cc1)N(CC(F)(F)F)c1ccc(Oc2nc(O)c3ccncc3n2)cc1

InChI Key InChIKey=PCTBZMTVWLMJTL-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 296189   

TargetLysine-specific demethylase 4C(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM296189(2-{4-[(4-isopropyl-phenyl)-(2,2,2-trifluoro- ethyl...)
Affinity DataIC50:  550nMAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate-format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM296189(2-{4-[(4-isopropyl-phenyl)-(2,2,2-trifluoro- ethyl...)
Affinity DataIC50:  550nMT: 2°CAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent