BDBM371353 1-(Cyclobutylmethyl)-N-[1-(fluoromethyl)cyclopropyl]-3-[(1-methylpyrazol-4-yl)methyl]-2,4-dioxo-quinazoline-6-sulfonamide::US10239843, Example 461
SMILES Cn1cc(Cn2c(=O)n(CC3CCC3)c3ccc(cc3c2=O)S(=O)(=O)NC2(CF)CC2)cn1
InChI Key InChIKey=MZANIXIFXUWZOT-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 371353
Affinity DataIC50: 39nMAssay Description:PARG In vitro assays were conducted in a total volume of 15 ul in a standard 384 well format. 5 ul of Human Full Length PARG (Produced internally by ...More data for this Ligand-Target Pair