BDBM416455 (R)-N-(2-(dimethylamino)-1-(4-(ethylsulfonyl)phenyl)ethyl)-1-ethyl-2-(4-(trifluoromethyl)phenoxy)-1H-benzo[d]imidazole-5-carboxamide::US10301261, Compound BE-10::US10829448, Compound BE-10

SMILES CCn1c(Oc2ccc(cc2)C(F)(F)F)nc2cc(ccc12)C(=O)N[C@@H](CN(C)C)c1ccc(cc1)S(=O)(=O)CC

InChI Key InChIKey=JZOPAHUJWUBNIB-VWLOTQADSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 416455   

TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Vitae Pharmaceuticals

US Patent
LigandPNGBDBM416455((R)-N-(2-(dimethylamino)-1-(4-(ethylsulfonyl)pheny...)
Affinity DataKi:  550nMAssay Description:Compounds described herein were tested for ability to bind to RORγ in a cell-free competition assay with commercially available radio-ligand (RL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Vitae Pharmaceuticals

US Patent
LigandPNGBDBM416455((R)-N-(2-(dimethylamino)-1-(4-(ethylsulfonyl)pheny...)
Affinity DataKi:  550nMAssay Description:Compounds described herein were tested for ability to bind to RORγ in a cell-free competition assay with commercially available radio-ligand (RL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent