BDBM464509 2-(((1s,4s)-4-((6-(4- methoxyphenyl)-3-oxo-5- phenyl-1,2,4-triazin-2(3H)- yl)methyl)cyclohexyl) methoxy)acetic acid::US10793529, Compound 69

SMILES COc1ccc(cc1)-c1nn(C[C@@H]2CC[C@H](COCC(O)=O)CC2)c(=O)nc1-c1ccccc1

InChI Key InChIKey=GWKZBHISORWCRW-KDURUIRLSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 464509   

TargetProstacyclin receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM464509(2-(((1s,4s)-4-((6-(4- methoxyphenyl)-3-oxo-5- phen...)
Affinity DataEC50:  8nMAssay Description:The HTRF® assay was carried out using a two-step protocol essentially according to the kit manufacturer's instructions, in 20 μL total volum...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent