BDBM464687 US10793563, Compound I-10::US10793563, Compound I-44::US10793563, Compound I-9

SMILES FC(F)(F)c1ccc2ncc(-c3ccnc(n3)N3CCOC(C3)c3cn[nH]c3)n2c1

InChI Key

Data  3 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 464687   

TargeteIF-2-alpha kinase GCN2(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM464687(US10793563, Compound I-10 | US10793563, Compound I...)
Affinity DataKi: <10nMAssay Description:An assay buffer containing GCN2 kinase and (RS)7 was prepared. 4.7 μL of this stock solution was placed per well of a black, low volume, 384-wel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargeteIF-2-alpha kinase GCN2(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM464687(US10793563, Compound I-10 | US10793563, Compound I...)
Affinity DataKi: <10nMAssay Description:An assay buffer containing GCN2 kinase and (RS)7 was prepared. 4.7 μL of this stock solution was placed per well of a black, low volume, 384-wel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargeteIF-2-alpha kinase GCN2(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM464687(US10793563, Compound I-10 | US10793563, Compound I...)
Affinity DataKi: <10nMAssay Description:An assay buffer containing GCN2 kinase and (RS)7 was prepared. 4.7 μL of this stock solution was placed per well of a black, low volume, 384-wel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent