BDBM468985 2-methyl-4-(2-methyl-1,1-dioxo-3H-1,2- benzothiazol-6-yl)isoquinolin-1-one::US10807982, Example 1
SMILES CN1Cc2ccc(cc2S1(=O)=O)-c1cn(C)c(=O)c2ccccc12
InChI Key InChIKey=PGBBIPXLGUYYEM-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 468985
Affinity DataIC50: 2.75E+3nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair