BDBM469045 5-(5-methoxy-2-methyl-1,1-dioxo-3H-1,2- benzothiazol-6-yl)-1,3-dimethylpyridin-2-one::US10807982, Example 3
SMILES COc1cc2CN(C)S(=O)(=O)c2cc1-c1cc(C)c(=O)n(C)c1
InChI Key InChIKey=GZDCYEJGWVUVLI-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469045
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair