BDBM469053 4-(5-methoxy-2-methyl-1,1-dioxo-3H-1,2- benzothiazol-6-yl)-2-methylisoquinolin-1-one::US10807982, Example 4
SMILES COc1cc2CN(C)S(=O)(=O)c2cc1-c1cn(C)c(=O)c2ccccc12
InChI Key InChIKey=DSJUYKKFXSJJDN-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469053
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair