BDBM469059 5-[5-(cyclopropylmethoxy)-2-methyl-1,1-dioxo- 3H-1,2-benzothiazol-6-yl]-1,3- dimethylpyridin-2-one::US10807982, Example 5
SMILES CN1Cc2cc(OCC3CC3)c(cc2S1(=O)=O)-c1cc(C)c(=O)n(C)c1
InChI Key InChIKey=JVQRZWYJOCYTAM-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469059
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair