BDBM469072 4-[5-(cyclopropylmethoxy)-2-methyl-1,1-dioxo- 3H-1,2-benzothiazol-6-yl]-2- methylisoquinolin-1-one::US10807982, Example 6
SMILES CN1Cc2cc(OCC3CC3)c(cc2S1(=O)=O)-c1cn(C)c(=O)c2ccccc12
InChI Key InChIKey=HCGHJQUBUGIUBL-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469072
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair