BDBM469095 5-[5-(cyclopropylmethoxy)-1-methylsulfonyl-2,3- dihydroindol-6-yl]-1,3-dimethylpyridin-2-one::US10807982, Example 15
SMILES Cc1cc(cn(C)c1=O)-c1cc2N(CCc2cc1OCC1CC1)S(C)(=O)=O
InChI Key InChIKey=GCADSKMWXUKYCI-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469095
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair