BDBM469102 5-[5-(cyclopropylmethoxy)-1-ethylsulfonyl-2,3- dihydroindol-6-yl]-1,3-dimethylpyridin-2-one::US10807982, Example 16
SMILES CCS(=O)(=O)N1CCc2cc(OCC3CC3)c(cc12)-c1cc(C)c(=O)n(C)c1
InChI Key InChIKey=DICYUGPHLWYCQT-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469102
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair