BDBM469119 N-[1-benzyl-6-(2-methyl-1-oxoisoquinolin-4-yl)- 2,3-dihydroindol-4-yl]methanesulfonamide::US10807982, Example 20
SMILES Cn1cc(-c2cc3N(Cc4ccccc4)CCc3c(NS(C)(=O)=O)c2)c2ccccc2c1=O
InChI Key InChIKey=PGDPQXDDOAIUHI-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469119
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair