BDBM469121 5-(2-ethyl-5-methylsulfonyl-1-benzofuran-7-yl)- 1,3-dimethylpyridin-2-one::US10807982, Example 21
SMILES CCc1cc2cc(cc(-c3cc(C)c(=O)n(C)c3)c2o1)S(C)(=O)=O
InChI Key InChIKey=MDSONSDVBTYUBR-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469121
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair