BDBM469124 N-[2-(1,5-dimethyl-6-oxopyridin-3-yl)-9-[(4- fluorophenyl)methyl]-8-methylpurin-6- yl]methanesulfonamide::US10807982, Example 22
SMILES Cc1nc2c(NS(C)(=O)=O)nc(nc2n1Cc1ccc(F)cc1)-c1cc(C)c(=O)n(C)c1
InChI Key InChIKey=MWMRNAUIHFFKQC-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469124
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair