BDBM469136 4-(2-cyclopropyl-5-ethylsulfonyl-1-benzofuran- 7-yl)-2-methylisoquinolin-1-one::US10807982, Example 24
SMILES Cn1cc(-c2cc(cc3cc(oc23)C2CC2)S(C)(=O)=O)c2ccccc2c1=O
InChI Key InChIKey=BMVGRYYCVHUNTL-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469136
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair