BDBM469146 2-methyl-4-(5-methylsulfonyl-2-phenyl-1- benzofuran-7-yl)isoquinolin-1-one::US10807982, Example 26
SMILES Cn1cc(-c2cc(cc3cc(oc23)-c2ccccc2)S(C)(=O)=O)c2ccccc2c1=O
InChI Key InChIKey=ADKKKJSPASMXOK-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469146
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair